Search Count: 32
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Crystal Structure Of Gmppnp Bound Kras-Y71H In Complex With Rbd Domain Of Craf(Raf1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2026-05-20 Classification: ONCOPROTEIN Ligands: GNP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-20
Ligands: GNP, MG
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Crystal Structure Of Gmppnp Bound Kras G12C In Complex With Cypa And Rmc-4791
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2026-05-20 Classification: ONCOPROTEIN Ligands: MG, GNP, A1CYT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-20
Ligands: MG, GNP, A1CYT
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Cryoem Structure Of Activated Craf/Mek/14-3-3 Complex With Nst-628
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
Ligands: A1AHE
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Activated Craf/Mek Heterotetramer From Focused Refinement Of Craf/Mek/14-3-3 Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
Ligands: A1AHE
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Crystal Structure Of Ksr1/Mek1 Complex Heterotetramer With Nst-628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, ANP, MG, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, ANP, MG, EDO, CL
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Crystal Structure Of Araf/Mek1 Complex With Nst-628 And A Raf Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, MG, ANP, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, MG, ANP, EDO, GOL
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Crystal Structure Of Braf/Mek1 Complex With Nst-628 And An Active Raf Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, ANP, MG, EDO, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, ANP, MG, EDO, TRS
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Crystal Structure Of Braf/Mek Complex With Nst-628 And Inactive Raf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: ANP, MG, A1AHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: ANP, MG, A1AHE
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Crystal Structure Of Craf/Mek1 Complex With Nst-628 And Inactive Raf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: ANP, MG, NI, ACT, EDO, A1AHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: ANP, MG, NI, ACT, EDO, A1AHE
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Crystal Structure Of Craf/Mek Complex With Nst-628 And Active Raf Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, ANP, MG
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Nanobret Tracer Tram-Bo Bound To A Ksr2-Mek1 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.23 Å Release Date: 2023-09-27 Classification: TRANSFERASE Ligands: ANP, U9F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-27
Ligands: ANP, U9F
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Cobimetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2020-10-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, EUI |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: ANP, MG, EUI
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Crystal Structure Of Ksr2:Mek1 In Complex With Adp
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ADP, MG
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Trametinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, QOM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, QOM
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Cobimetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKD |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKD
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Crystal Structure Of Ksr2:Mek1 In Complex With Anp-Pnp, And Allosteric Mek Inhibitor Selumetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, 3EW |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, 3EW
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Pd0325901
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, 4BM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, 4BM
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Aps-9-95-1
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.36 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKG
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Trametinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, QOM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, QOM
