Search Count: 6
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Cyanofluorophenylacetamides As Orally Efficacious Thrombin Inhibitors
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2009-02-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DKK |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: DKK
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Glycogen Synthase Kinase-3 Beta In Complex With Bis-(Indole)Maleimide Pyridinophane Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-02-19 Classification: TRANSFERASE Ligands: BIM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-19
Ligands: BIM
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X-Ray Structure Of Fxa In Complex With 7-Fluoroindazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-01-29 Classification: HYDROLASE Ligands: JNJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: JNJ
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Discovery Of Potent, Orally Active, Nonpeptide Inhibitors Of Human Mast Cell Chymase By Using Structure-Based Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2007-06-12 Classification: HYDROLASE Ligands: DRX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-06-12
Ligands: DRX
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A Dual Inhibitor Of The Leukocyte Proteases Cathepsin G And Chymase With Therapeutic Efficacy In Animals Models Of Inflammation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: NAG, SO4, CO, OHH, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: NAG, SO4, CO, OHH, MES
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A Dual Inhibitor Of The Leukocyte Proteases Cathepsin G And Chymase With Therapeutic Efficacy In Animals Models Of Inflammation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: SO4, OHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: SO4, OHH
