Search Count: 37
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-05-28 Classification: HYDROLASE Ligands: CA, A1A8O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1A8O
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Inhibiting Peptidylarginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, A1BZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1BZK
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1A9P, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1A9P, 3YZ
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Discovery Of A High Affinity Inhibitor Of Cgas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.23 Å Release Date: 2018-12-19 Classification: transferase/transferase inhibitor Ligands: ZN, KHM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: ZN, KHM
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Human Pim1 Kinase In Complex With Compound 12B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2018-03-21 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: EDO, MVG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: EDO, MVG, SO4
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Discovery Of A High Affinity Inhibitor Of Cgas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2017-09-27 Classification: transferase/transferase inhibitor Ligands: ZN, 8ZM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 8ZM
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With 2',2'-Cgamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 1YC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 1YC
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With 2',3'-Cgamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, SO4, 1SY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, SO4, 1SY
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With 2',5'-Gpap
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 9BG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 9BG
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With 3',3'-Cdimp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 9B7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 9B7
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With 3',3'-Cdump
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 9BJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 9BJ
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With 3',3'-Cgamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 4BW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 4BW
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound F2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 9BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 9BS
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound F3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 9BV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 9BV, SO4
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Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound F1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2017-09-27 Classification: TRANSFERASE Ligands: ZN, 9BY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: ZN, 9BY
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Structure Of Human Polycomb Repressive Complex 2 (Prc2) With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.47 Å Release Date: 2017-02-22 Classification: Transferase/Inhibitor Ligands: ZN, 74D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 74D
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Smyd2 In Complex With Az370
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2016-12-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, BU3, 6T1, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: SAM, BU3, 6T1, ZN
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Smyd2 In Complex With Az378
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-12-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: SAM, ZN
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Smyd2 In Complex With Az931
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2016-12-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 6TM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: SAM, 6TM, ZN
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Smyd2 In Complex With Az506
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2016-12-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, BU3, NA, 6TL, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: SAM, BU3, NA, 6TL, ZN