Search Count: 13
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Crystal Structure Of Au-15330 In Complex With The Bromodomain Of Human Brm (Smarca2) And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2025-10-08 Classification: TRANSCRIPTION Ligands: A1BNT, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-08
Ligands: A1BNT, EDO, GOL
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Crystal Structure Of Prt3789 In Complex With The Bromodomain Of Human Brg1 (Smarca4) And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-10-01 Classification: TRANSCRIPTION Ligands: A1BB4, GOL, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: A1BB4, GOL, EDO, CL
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Crystal Structure Of Prt3789 In Complex With The Bromodomain Of Human Brm (Smarca2) And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2025-10-01 Classification: TRANSCRIPTION Ligands: A1BB4, CIT, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: A1BB4, CIT, ACT
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Crystal Structure Of The Bromodomain Of Human Brm (Smarca2) In Complex With A Smarca-Bd Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2025-10-01 Classification: TRANSCRIPTION Ligands: A1BB5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: A1BB5, ZN
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Crystal Structure Of Catalytic Domain Of Tace With 2-(2-Aminothiazol-4-Yl)Pyrrolidine-Based Tartrate Diamides
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2011-04-20 Classification: hydrolase/hydrolase inhibitor Ligands: IPA, INN, ZN, CA, 786 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: IPA, INN, ZN, CA, 786
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X-Ray Crystal Structure Of Compound 70 Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2010-12-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: C70 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-08
Ligands: C70
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X-Ray Crystal Structure Of Compound 2A Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2010-12-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: C72, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-08
Ligands: C72, GOL
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X-Ray Crystal Structure Of Compound 1 Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2010-12-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: C73, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-08
Ligands: C73, GOL
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Crystal Structure Of Catalytic Domain Of Tace With Benzimidazolyl-Thienyl-Tartrate Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-07-28 Classification: HYDROLASE Ligands: ZN, 50X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: ZN, 50X
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Crystal Structure Of Catalytic Domain Of Tace With Hydantoin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, INN, IPA, Z94 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ZN, INN, IPA, Z94
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Crystal Structure Of Catalytic Domain Of Tace With The First Hydantoin Inhibitor Occupying The S1' Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 724 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ZN, 724
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Crystal Structure Of Catalytic Domain Of Tace With Tartrate-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: ZN, INN, 403 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: ZN, INN, 403
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Crystal Structure Of Catalytic Domain Of Tace With Phenyl-Pyrrolidinyl-Tartrate Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: ZN, INN, IPA, Z59 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: ZN, INN, IPA, Z59