Search Count: 38
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Structure Of The Human Ddb1-Dda1-Dcaf15 E3 Ubiquitin Ligase Bound To Rbm39 And Sulfonamide E7820
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-09-18 Classification: LIGASE Ligands: EPE, O6M, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-18
Ligands: EPE, O6M, ZN
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Jak3 With Cyanamide Cp10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G4V
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Jak3 With Cyanamide Cp23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G54 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G54
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Jak3 With Cyanamide Cp34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G4Y
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Jak3 With Cyanamide Cp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-11-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HB4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: HB4, SO4
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Jak3 With Covalent Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KU
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Jak3 With Covalent Inhibitor 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KV, SO4
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Jak3 With Covalent Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KX
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Crystal Structure Of Pt2385 Bound To Hif2A-B*:Arnt-B* Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-09-21 Classification: TRANSCRIPTION Ligands: 79A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 79A
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Crystal Structure Of Itk In Complex With Compound 1 [4-(Carbamoylamino)-1-(Naphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Y
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Crystal Structure Of Itk In Complex With Compound 5 {4-(Carbamoylamino)-1-(7-Methoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide}
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Z
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Crystal Structure Of Itk In Complex With Compound 7 [4-(Carbamoylamino)-1-(7-Ethoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1YZ
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Crystal Structure Of Itk In Complex With Compound 8 [4-(Carbamoylamino)-1-(7-Propoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1E0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1E0
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide] And Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS, ADP
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Crystal Structure Of Itk In Complex With Compound 52
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2012-11-14 Classification: transferase/transferase inhibitor Ligands: 18R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 18R
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Crystal Structure Of Itk In Complext With Compound 40
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2012-11-14 Classification: transferase/transferase inhibitor Ligands: 13L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 13L
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Crystal Structure Of Itk In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2012-11-14 Classification: transferase/transferase inhibitor Ligands: 13J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 13J
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Amcase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-08-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3RM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-24
Ligands: 3RM
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Amcase In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-08-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RM8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-24
Ligands: RM8