Search Count: 19
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Human Gkrp Bound To Amg2882 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WY, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3295 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0265 (N-[(R)-(2-Chlorophenyl){7-[4-(2-Hydroxypropan-2-Yl) Pyridin-2-Yl]-1-Benzothiophen-2-Yl}Methyl]Cyclopropanesulfonamide) And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 2Y6, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 2Y6, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-2526 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-08 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TE, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 2TE, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0771 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TF, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TF, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-2668
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TG, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TG, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3227 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TJ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TJ, S6P, IOD, GOL, SO4
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Gkrp Bound To Amg0556 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UW, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UW, S6P, IOD, GOL, SO4
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Gkrp Bound To Amg-0471 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5112 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UY, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg5106 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-23 Classification: CARBOHYDRATE BINDING PROTEIN Ligands: 2TO, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 2TO, S6P, IOD, GOL, SO4
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Human Gkrp Complexed To Amg-3969 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG9, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG9, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5980 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG0, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG0, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-6861 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-03-12 Classification: SUGAR BINDING PROTEIN Ligands: 2EU, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-12
Ligands: 2EU, S6P, IOD, GOL, SO4
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Human Gkrp Complexed To Amg-1694 [(2R)-1,1,1-Trifluoro-2-{4-[(2S)-2-{[(3S)-3-Methylmorpholin-4-Yl]Methyl}-4-(Thiophen-2-Ylsulfonyl)Piperazin-1-Yl]Phenyl}Propan-2-Ol] And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-11-20 Classification: Carbohydrate Binding protein Ligands: IOD, S6P, 1YY, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: IOD, S6P, 1YY, GOL, SO4
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Cocrystal Structure Of Unphosphorylated Igf With Pyrimidine 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 01P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: 01P
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Further Studies With The 2-Amino-1,3-Thiazol-4(5H)-One Class Of 11-Hydroxysteroid Dehydrogenase Type 1 (11-Hsd1) Inhibitors: Reducing Pregnane X Receptor (Pxr) Activity And Exploring Activity In A Monkey Pharmacodynamic Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2008-11-11 Classification: OXIDOREDUCTASE Ligands: NDP, 352 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-11
Ligands: NDP, 352
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase(Hsd1) In Complex With Nadp And Thiazolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2008-06-10 Classification: OXIDOREDUCTASE Ligands: NAP, A21 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: NAP, A21
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The Discovery Of 2-Anilinothiazolones As 11Beta-Hsd1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2008-01-15 Classification: OXIDOREDUCTASE Ligands: ZMG, NDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: ZMG, NDP