Search Count: 24
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Cecr2 In Complex With Cpd6 (6-Allyl-N,2-Dimethyl-7-Oxo-N-(1-(1-Phenylethyl)Piperidin-4-Yl)-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-06-14 Classification: Transcription/Inhibitor Ligands: SO4, 96V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-14
Ligands: SO4, 96V
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Structure Of Human Polycomb Repressive Complex 2 (Prc2) With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.47 Å Release Date: 2017-02-22 Classification: Transferase/Inhibitor Ligands: ZN, 74D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 74D
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Kdm4C Bound To Pyrazolo-Pyrimidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-08-17 Classification: OXIDOREDUCTASE Ligands: FE2, ZN, 6X9, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: FE2, ZN, 6X9, CL
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Crystal Structure Of Kdm5A In Complex With A Naphthyridone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2016-08-10 Classification: Oxidoreductase/Inhibitor Ligands: NI, ZN, 6QN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: NI, ZN, 6QN
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Structure Of Histone Lysine Demethylase Kdm5A In Complex With Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Inhibitor Ligands: NI, ZN, 50P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NI, ZN, 50P
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 986, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 986, EDO
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi703
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING Ligands: 58N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 58N
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02773986
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: SCN, 68Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: SCN, 68Y
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02778174
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: EDO, SCN, 69A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: EDO, SCN, 69A
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02857790
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: ACT, CA, 69B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ACT, CA, 69B
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Cbp In Complex With Cpd23 ((R)-6-(3-(Benzyloxy)Phenyl)-4-Methyl-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69F, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69F, B3P, EDO, NA, PEG
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Cbp In Complex With Cpd637 ((R)-4-Methyl-6-(1-Methyl-3-(1-Methyl-1H-Pyrazol-4-Yl)-1H-Indazol-5-Yl)-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69E, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69E, B3P, EDO, NA, PEG
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Cpi-0610
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2016-02-10 Classification: TRANSCRIPTION Ligands: 62G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 62G
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Benzoisoxazoloazepine 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-02-10 Classification: TRANSCRIPTION Ligands: 62V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 62V
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Discovery Of Benzotriazolo Diazepines As Orally-Active Inhibitors Of Bet Bromodomains: Crystal Structure Of Brd4 With Cpi-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2015-11-11 Classification: SIGNALING PROTEIN Ligands: FMT, 3X0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: FMT, 3X0
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Benzotriazolo-Diazepine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2015-04-08 Classification: TRANSCRIPTION Ligands: 558 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 558
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Crystal Structure Of The First Bromodomain Of Human Brd4 With Benzotriazolo-Diazepine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2015-04-08 Classification: SIGNALING PROTEIN Ligands: 559 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 559
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The Crystal Structure Of Pcsk9 In Complex With 1D05 Fab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-11-03 Classification: HYDROLASE/ANTIBODY Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-03
Ligands: CA
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Wt Pcsk9-Deltac Bound To Wt Egf-A Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA
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Wt Pcsk9-Deltac Bound To Egf-A H306Y Mutant Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA