Search Count: 37
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1E
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: SO4, A1A1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: SO4, A1A1D
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1C
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1B, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1B, CL
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1A
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-[6-Chloro-4-(9-Methyl-1-Oxa-4,9-Diazaspiro[5.5]Undec-4-Yl)-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl]Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2023-04-05 Classification: TRANSFERASE Ligands: XXF, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF, SO4
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(3R,5S)-3-Amino-5-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
 |
Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(2S,5R)-5-Amino-2-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3O
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Pkceta Kinase Domain In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: XXF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF
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Pkceta Kinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
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Crystal Structure Of Nonphosphorylated, Hpk1 Kinase Domain In Complex With Sunitinib In The Inactive State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
 |
Crystal Structure Of Diphosphorylated Hpk1 Kinase Domain In Complex With Sunitinib In The Active State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2019-05-01 Classification: SIGNALING PROTEIN Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Sunitinib In The Inactive State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
 |
Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 10B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: FKY
 |
Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 13B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GO7
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 19.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GOD
 |
Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: GXA
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Structure Of The Ptk6 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-06-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
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Structure Of The Ptk6 Kinase Domain Bound To A Type I Inhibitor (3-Fluoro-4-{[6-Methyl-3-(1H-Pyrazol-4-Yl)Imidazo[1,2-A]Pyrazin-8-Yl]Amino}Phenyl)(Morpholin-4-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-06-20 Classification: Transferase/Transferase Inhibitor Ligands: FLJ, ACT, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-20
Ligands: FLJ, ACT, K
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Structure Of The Ptk6 Kinase Domain Bound To A Type Ii Inhibitor 2-{[(3R,4S)-3-Fluoro-1-{[4-(Trifluoromethoxy)Phenyl]Acetyl}Piperidin-4-Yl]Oxy}-5-(1-Methyl-1H-Imidazol-4-Yl)Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2018-06-20 Classification: Transferase/Transferase Inhibitor Ligands: FKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-20
Ligands: FKY