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Search Count: 18

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9ETQ image
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)

9ETR image
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574

8BSK image
Human Gls In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2023-01-18
Classification: HYDROLASE
Ligands: SO4, 04A

8BSL image
Human Gls In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2023-01-18
Classification: HYDROLASE
Ligands: R90

8BSM image
Human Gls In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.78 Å Release Date: 2023-01-18
Classification: HYDROLASE
Ligands: SO4, 5XX

8BSN image
Human Gls In Complex With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2023-01-18
Classification: HYDROLASE
Ligands: SO4, R0C

7ONR image
Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKW, SO4

7ONS image
Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKT, SO4

7ONT image
Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKQ, SO4

4D2R image
Human Igf In Complex With A Dyrk1B Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: CL, DYK

4D2S image
Human Ttk In Complex With A Dyrk1B Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: DYK

5AJV image
Human Pfkfb3 In Complex With An Indole Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.01 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: PO4, 8R2, FDP

5AJW image
Human Pfkfb3 In Complex With An Indole Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: PHS, PO4, F6P, S6L

5AJX image
Human Pfkfb3 In Complex With An Indole Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.58 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: PHS, PO4, F6P, FD9

5AJY image
Human Pfkfb3 In Complex With An Indole Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.37 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: PHS, PO4, F6P, 87T

5AJZ image
Human Pfkfb3 In Complex With An Indole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: PHS, F6P, PO4, MJP

5AK0 image
Human Pfkfb3 In Complex With An Indole Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2015-04-22
Classification: TRANSFERASE
Ligands: PHS, PO4, F6P, 8V1

1IK9 image
Crystal Structure Of A Xrcc4-Dna Ligase Iv Complex
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