Search Count: 35
![]() |
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
![]() |
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
![]() |
Human Gls In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, 04A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, 04A
![]() |
Human Gls In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: R90 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: R90
![]() |
Human Gls In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, 5XX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, 5XX
![]() |
Human Gls In Complex With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, R0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, R0C
![]() |
Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
![]() |
Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
![]() |
Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
![]() |
Human Pfkfb3 In Complex With A Pyrrolopyrimidone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-01-20 Classification: TRANSFERASE Ligands: PO4, PHS, F6P, BKI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: PO4, PHS, F6P, BKI
![]() |
Human Pfkfb3 In Complex With A Pyrrolopyrimidone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.24 Å Release Date: 2016-01-20 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, BKE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: PHS, PO4, F6P, BKE
![]() |
Human Pfkfb3 In Complex With A Pyrrolopyrimidone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.16 Å Release Date: 2016-01-20 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, BKS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: PHS, PO4, F6P, BKS
![]() |
Human Pfkfb3 In Complex With A Pyrrolopyrimidone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2016-01-20 Classification: TRANSFERASE Ligands: PO4, PHS, F6P, BKV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: PO4, PHS, F6P, BKV
![]() |
Human Igf In Complex With A Dyrk1B Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: CL, DYK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: CL, DYK
![]() |
Human Ttk In Complex With A Dyrk1B Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: DYK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: DYK
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PO4, 8R2, FDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PO4, 8R2, FDP
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, S6L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, S6L
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, FD9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, FD9
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 87T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 87T
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, F6P, PO4, MJP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, F6P, PO4, MJP
