Search Count: 13
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Crystal Structure Of Menin In Complex With Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVE
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Crystal Structure Of Menin In Complex With Inhibitor Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVF, K, EPE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVF, K, EPE, SO4
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Crystal Structure Of Menin In Complex With Inhibitor Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVG
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Pf-07284892
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-05-29 Classification: HYDROLASE/INHIBITOR Ligands: A1AQ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: A1AQ1
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Inhibitor Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2024-01-03 Classification: HYDROLASE/INHIBITOR Ligands: W8I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: W8I
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Inhibitor Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-01-03 Classification: HYDROLASE/INHIBITOR Ligands: WAB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: WAB
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Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, M1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, M1R
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Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, QH4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, QH4
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Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, M1X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, M1X
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: NI, 1M4
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: NI, 1M5
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: NI, 1M6
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: NI, 1M7
