Search Count: 21
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With (2S)-2-((3R)-3-Acetamido-3-Isobutyl-2-Oxo-1-Pyrrolidinyl)-N-((1S,2R)-1-(3,5-Difluorobenzyl)-2-Hydroxy-2-(1,2,3,4-Tetrahydro-3-Isoquinolinyl)Ethyl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2011-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-07
Ligands: PB8
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With (2S)-2-((3S)-3-(Acetylamino)-3-(Butan-2-Yl)-2-Oxopyrrolidin-1-Yl)-N-((2S,3R)-3-Hydroxy-4-((3-Methoxybenzyl)Amino)-1-Phenylbutan-2-Yl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB7, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PB7, IOD
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Crystal Structure Of Protein Tyrosine Phosphatase 1B In Complex With An Isothiazolidinone-Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: IZ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: IZ1
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Crystal Structure Of Protein Tyrosine Phosphatase 1B In Complex With An Isothiazolidinone-Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: IZ2, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: IZ2, MG
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Crystal Structure Of Protein Tyrosine Phosphatase 1B In Complex With An Isothiazolidinone-Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: IZ3, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: IZ3, MG
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Crystal Structure Of Protein Tyrosine Phosphatase 1B In Complex With An Isothiazolidinone-Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: IZ4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: IZ4, MG
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Crystal Structure Of Protein Tyrosine Phosphatase 1B In Complex With An Isothiazolidinone-Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: IZ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: IZ5
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Structural Insights Into The Design Of Nonpeptidic Isothiazolidinone- Containing Inhibitors Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2006-09-27 Classification: HYDROLASE Ligands: DFJ, SO4, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-27
Ligands: DFJ, SO4, BOG
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Structural Insights Into The Design Of Nonpeptidic Isothiazolidinone- Containing Inhibitors Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-09-27 Classification: HYDROLASE Ligands: F32, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-27
Ligands: F32, MG
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Structural Insights Into The Design Of Nonpeptidic Isothiazolidinone- Containing Inhibitors Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-09-27 Classification: HYDROLASE Ligands: IZE, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-27
Ligands: IZE, MG, GOL
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Structural Insights Into The Design Of Nonpeptidic Isothiazolidinone- Containing Inhibitors Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2006-09-27 Classification: HYDROLASE Ligands: CA, IZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-27
Ligands: CA, IZB
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Structural Insights Into The Design Of Nonpeptidic Isothiazolidinone- Containing Inhibitors Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-09-27 Classification: HYDROLASE Ligands: IZF, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-27
Ligands: IZF, MG
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Structure Of Protein Tyrosine Phosphatase 1B (P212121)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: MPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: MPD
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Structure Of Protein Tyrosine Phosphatase 1B (C2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: CA
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Structural Basis For Inhibition Of Protein Tyrosine Phosphatase 1B By Isothiazolidinone Heterocyclic Phosphonate Mimetics
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: IZD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: IZD
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Structural Basis For Inhibition Of Protein Tyrosine Phosphatase 1B By Isothiazolidinone Heterocyclic Phosphonate Mimetics
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: F16, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: F16, MG
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Structural Basis For Inhibition Of Protein Tyrosine Phosphatase 1B By Isothiazolidinone Heterocyclic Phosphonate Mimetics
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: F20 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: F20
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Structural Basis For Inhibition Of Protein Tyrosine Phosphatase 1B By Isothiazolidinone Heterocyclic Phosphonate Mimetics
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: F17, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: F17, BOG
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Structural Basis For Inhibition Of Protein Tyrosine Phosphatase 1B By Isothiazolidinone Heterocyclic Phosphonate Mimetics
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-08-17 Classification: HYDROLASE Ligands: DFM, SO4, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-17
Ligands: DFM, SO4, BOG
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Structure Of Signal Transduction Protein, Nmr, Minimized Average Structure
Organism: Gallus gallus
Method: SOLUTION NMR Release Date: 1997-01-27 Classification: COMPLEX (TRANSFERASE/PEPTIDE) |
Organism: Gallus gallus
Method: SOLUTION NMR
Release Date: 1997-01-27
