Search Count: 22
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Crystal Structure Of Fxa In Complex With 4,4-Disubstituted Pyrrolidine-1,2-Dicarboxamide Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-04-07 Classification: HYDROLASE Ligands: CA, L1C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: CA, L1C
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Crystal Structure Of Fxa In Complex With 4,4-Disubstituted Pyrrolidine-1,2-Dicarboxamide Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2009-04-07 Classification: HYDROLASE Ligands: L1D, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: L1D, CA
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An Orally Efficacious Factor Xa Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-03-25 Classification: BLOOD CLOTTING Ligands: CA, 230 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-25
Ligands: CA, 230
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Factor Xa Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2007-08-14 Classification: BLOOD CLOTTING Ligands: CA, 237 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-14
Ligands: CA, 237
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The Discovery Of Glycine And Related Amino Acid-Based Factor Xa Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2007-08-14 Classification: HYDROLASE Ligands: CA, FXI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-14
Ligands: CA, FXI
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Crystal Structure Of Human Renin Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2006-12-05 Classification: HYDROLASE Ligands: LIY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-05
Ligands: LIY
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Crystal Structure Of Human Renin Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2006-12-05 Classification: HYDROLASE Ligands: LIX, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-05
Ligands: LIX, CIT
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Crystal Structure Of Human Renin Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-11-14 Classification: HYDROLASE Ligands: 7IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-14
Ligands: 7IG
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Crystal Structure Of Factor Vii.Stf Complexed With Pd0297121
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2006-10-18 Classification: HYDROLASE Ligands: CA, GIL, GLC, FUC, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-10-18
Ligands: CA, GIL, GLC, FUC, NAG
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Crystal Structure Of A Ternary Complex Of Factor Viia/Tissue Factor And 2-[[6-[3-(Aminoiminomethyl)Phenoxy]-3,5-Difluro-4-[(1-Methyl-3-Phenylpropyl)Amino]-2-Pyridinyl]Oxy]-Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2006-08-01 Classification: HYDROLASE Ligands: CA, CAC, 03R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-01
Ligands: CA, CAC, 03R
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-06-20 Classification: HYDROLASE Ligands: L1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-20
Ligands: L1A
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: PZ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: PZ1
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 1IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 1IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 2IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 2IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 3IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 3IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 4IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 4IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 5IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 5IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: L1B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: L1B
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 6IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 6IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: 7IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: 7IG
