Search Count: 28
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Crystal Structure Of Htead2 Bound To A Methoxypyridine Lipid Pocket Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-08-16 Classification: TRANSCRIPTION/INHIBITOR Ligands: TRS, Y2S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: TRS, Y2S
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Tead2 Bound To Gne-7883
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: TRS, KUR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: TRS, KUR
 |
Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: KUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: KUI
 |
Tead2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: KTF, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: KTF, TRS
 |
Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: 799 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: 799
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3W
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3R
 |
Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3N
 |
Crystal Structure Of Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-06-24 Classification: Transcription/Transcription Inhibitor Ligands: GOL, QSJ, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: GOL, QSJ, TRS
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Crystal Structure Of Tead2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2020-06-24 Classification: TRANSCRIPTION/INHIBITOR Ligands: QLV, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: QLV, TRS
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Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
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Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
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Egfr Kinase Domain Mutant "Tmlr" With 3-Azetidinyl Azaindazole Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60E
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Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 2: 4-[2-(4-Chlorophenyl)Ethylamino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q2
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Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 19: 4-[(2-Azanylpyrimidin-4-Yl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 5Q3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5Q3
 |
Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 13: 4-[(2-Methoxyphenyl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 5Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5Q4
 |
Egfr Kinase Domain With Pyridone Compound 13: 4-[(2-Methoxyphenyl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q4
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YV
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YW
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4YX