Search Count: 14
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Crystal Structure Of The Mertk Kinase Domain With Sa4488
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-10-09 Classification: TRANSFERASE Ligands: A1APF, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APF, CL
 |
Cdk2 With Compound 14 Inhibitor With Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-07-07 Classification: SIGNALING PROTEIN, Transferase/Inhibitor Ligands: YOS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: YOS
 |
Discovery Of Spirohydantoins As Selective, Orally Bioavailable Inhibitors Of P300/Cbp Histone Acetyltransferases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2021-03-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Y2P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-17
Ligands: Y2P
 |
Crystal Structure Of Human Nampt With Fragment 2: 2-[(2-Fluorophenyl)Amino]-6-Propylpyrimidin-4(3H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-01-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: AQ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-10
Ligands: AQ1
 |
Crystal Structure Of Human Nampt With Fragment 5: (3E)-3-[(Phenylamino)Methylidene]Oxan-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2018-01-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: AOY, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-10
Ligands: AOY, SO4
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Crystal Structure Of Human Nampt With A-1293201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: 7T7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7T7, SO4
 |
Crystal Structure Of Human Nampt With A-1326133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 7TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: SO4, 7TA
 |
Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HY
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HV
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Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(2-Methoxyphenyl)Methyl]-N,N-Dimethyl-4-(1-Methylindol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING, INHIBITOR Ligands: LQD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: LQD
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Polycomb Protein Eed In Complex With Inhibitor: 2-[4-(4-{(3S,4R)-4-(Dimethylamino)-1-[(2-Fluoro-6-Methylphenyl)Methyl]Pyrrolidin-3-Yl}Phenyl)-1H-Pyrazol-1-Yl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING, INHIBITOR Ligands: 7XG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 7XG
 |
Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(2-Bromo-6-Fluorophenyl)Methyl]-N,N-Dimethyl-4-(1-Methyl-1H-Indol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: 82D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 82D
 |
Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(1S)-7-Fluoro-2,3-Dihydro-1H-Inden-1-Yl]-N,N-Dimethyl-4-(1-Methyl-1H-Indol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: 82G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 82G
 |
Egfr Kinase Domain Complexed With An Imidazo[2,1-B]Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ITI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-02
Ligands: ITI