Search Count: 21
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Mtb Guab Dcbs In Complex With Inhibitor G1
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-27 Classification: OXIDOREDUCTASE Ligands: IMP, VOA, SO4 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: IMP, VOA, SO4
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Mtb Guab Dcbs In Complex With Inhibitor Compound 5
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-27 Classification: OXIDOREDUCTASE Ligands: IMP, A1A3K |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: IMP, A1A3K
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Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
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Crystal Structure Of Ire1A In Complex With G-6904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N8S, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N8S, EPE
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Crystal Structure Of Ire1 In Complex With G-3053
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-04-21 Classification: TRANSFERASE/INHIBITOR Ligands: N97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N97
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Crystal Structure Of Ire1A In Complex With G-4100
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
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Structure Of Unphosphorylated Ire1 In Complex With G-1749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJG
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Structure Of Unphosphorylated Ire1 In Complex With G-7658
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJM
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Structure Of Apo Unphosphorylated Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Apo Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Ire1 In Complex With G-0701
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJV
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Structure Of Unphosphorylated Human Ire1 Bound To G-9807
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2020-12-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SJS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJS
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Crebbp Bromodomain In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2018-02-21 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 9U4
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Crebbp Bromodomain In Complex With Cpd6 (Methyl 1H-Indole-3-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: DMS, C2Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: DMS, C2Y
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Crebbp Bromodomain In Complex With Cpd16 (5-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1H-Indole-3-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: C3J, EDO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: C3J, EDO, NA
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Crebbp Bromodomain In Complex With Cpd17 (5-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-3-Methylbenzo[D]Thiazol-2(3H)-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: C3V, SO4, DMS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: C3V, SO4, DMS, GOL
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Usp7 In Complex With Gne6640 (4-(2-Amino-4-Ethyl-5-(1H-Indazol-5-Yl)Pyridin-3-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JM
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Usp7 In Complex With Gne6776 (6'-Amino-4'-Ethyl-5'-(4-Hydroxyphenyl)-N-Methyl-[3,3'-Bipyridine]-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JP
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Crystal Structure Of Cdk8:Cyclin C Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-02-10 Classification: Transcription/Transferase/Inhibitor Ligands: EDO, FMT, 50R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: EDO, FMT, 50R
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Human Nav1.7-Vsd4-Navab In Complex With Gx-936.
Organism: Arcobacter butzleri, homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.53 Å Release Date: 2015-12-23 Classification: METAL TRANSPORT Ligands: PX4, 5P2 |
Organism: Arcobacter butzleri, homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-23
Ligands: PX4, 5P2