Search Count: 20
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The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7W |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: H7W
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The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With An Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7Z |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: H7Z
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Structure Of Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: FSU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: FSU
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Structure Of Human Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: D7N
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Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: SO4, GOL, FSU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: SO4, GOL, FSU
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Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: D7N, SO4
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Novel Pyrrole Carboxamide Inhibitors Of Jak2 As Potential Treatment Of Myeloproliferative Disorders
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-04-29 Classification: TRANSFERASE Ligands: QUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: QUP
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B-Raf Kinase V600E Mutant In Complex With A Diarylthiazole B-Raf Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: CQE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: CQE
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: GOL, VVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: GOL, VVQ
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: 953, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 953, GOL
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: BJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: BJG
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Structure Of Hsp90 With Nms-E973 Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-05-29 Classification: CHAPERONE Ligands: 9UN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 9UN
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Optimisation Of 6,6-Dimethyl Pyrrolo 3,4-C Pyrazoles: Identification Of Pha-793887, A Potent Cdk Inhibitor Suitable For Intravenous Dosing
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-02-23 Classification: CELL CYCLE Ligands: SO4, 889 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: SO4, 889
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Structure Of Cdk2-Cyclin A With A Pyrazolo(4,3-H) Quinazoline-3- Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-02-23 Classification: TRANSFERASE Ligands: WXV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: WXV, SO4
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Structure Of Cdk2-Cyclin A With Pha-848125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P48, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P48, SO4
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Structure Of Cdk2-Cyclin A Complexed With 8-Anilino-1-Methyl-4,5-Dihydro- 1H-Pyrazolo[4,3-H] Quinazoline-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P49, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P49, SO4
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Structure Of Cdk2-Cyclin A With Pha-630529
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-12-08 Classification: TRANSFERASE Ligands: 529, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-12-08
Ligands: 529, SO4
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Structure Of Cdk2-Cyclin A With Pha-533514
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2005-11-23 Classification: TRANSFERASE Ligands: SO4, 514 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-23
Ligands: SO4, 514
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Structure Of Cdk2 Complexed With Pnu-181227
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2004-06-17 Classification: TRANSFERASE Ligands: N5B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-06-17
Ligands: N5B
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Structure Of Cdk2/Cyclin A With Pnu-292137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2004-06-10 Classification: TRANSFERASE Ligands: SO4, 292 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-06-10
Ligands: SO4, 292
