Search Count: 40
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Crystal Structure Of Jak2 Jh1 With Type Ii Inhibitor Yliu-04-105-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2023-06-21 Classification: TRANSFERASE/INHIBITOR Ligands: I6C, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-21
Ligands: I6C, GOL
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZF
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZL
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZO, MG
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZR
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: G0U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: G0U
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: G5C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: G5C
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Crystal Structure Of Egfr 696-1022 Wt In Complex With Azd9291 Prepared By Cocrystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: YY3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: YY3, CL
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Crystal Structure Of Egfr 696-1022 L858R In Complex With Azd9291
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2020-04-22 Classification: TRANSFERASE Ligands: YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: YY3
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Crystal Structure Of Egfr 696-1022 T790M In Complex With Azd9291 Prepared By Co-Crystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2020-04-22 Classification: TRANSFERASE Ligands: YY3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: YY3, CL
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Crystal Structure Of Egfr 696-1022 T790M In Complex With Azd9291 Prepared By Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2020-04-22 Classification: TRANSFERASE Ligands: YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: YY3
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Irak4 In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2019-02-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI, SO4, CO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: 0LI, SO4, CO
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Irak4 In Complex With A Type Ii Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2019-02-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J8A, SO4, CO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: J8A, SO4, CO
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Crystal Structure Of The Unphosphorylated Irak4 Kinase Domain Bound To A Type I Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-02-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J87 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-13
Ligands: J87
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Crystal Structure Of The Unphosphorylated Irak4 Kinase Domain Bound To A Type I Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2019-02-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DL1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-13
Ligands: DL1
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Crystal Structure Of The Inactive Unphosphorylated Irak4 Kinase Domain Bound To Amp-Pnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-02-13 Classification: SIGNALING PROTEIN Ligands: ANP, SO4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-13
Ligands: ANP, SO4, MG
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Crystal Structure Of Ack1 With Compound 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2018-09-26 Classification: TRANSFERASE Ligands: 9KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: 9KO
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Dyrk1A In Complex With Xmd7-117
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: B5T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: B5T
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Dyrk1A In Complex With Hg-8-60-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: B5Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: B5Z
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Dyrk1A In Complex With Xmd8-49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: B6B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: B6B
