Search Count: 30
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Human Gkrp Bound To Amg2882 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WY, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3295 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0696 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WZ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WZ, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0265 (N-[(R)-(2-Chlorophenyl){7-[4-(2-Hydroxypropan-2-Yl) Pyridin-2-Yl]-1-Benzothiophen-2-Yl}Methyl]Cyclopropanesulfonamide) And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 2Y6, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 2Y6, S6P, IOD, GOL, SO4
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Crystal Structure Of 2-(3-Alkoxy-1-Azetidinyl) Quinolines As Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: SO4, GOL, 35E, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, GOL, 35E, ZN
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2-(3-Alkoxy-1-Azetidinyl) Quinolines As Novel Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, GOL, 35D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: ZN, SO4, GOL, 35D
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Human Gkrp Bound To Amg-2526 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-08 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TE, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 2TE, S6P, IOD, GOL, SO4
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Crystal Structure Of Pde10A With A Novel Imidazo[4,5-B]Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2014-10-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1IS, 1IR, ZN, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-01
Ligands: 1IS, 1IR, ZN, SO4, GOL
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Crystal Structure Of Pde10A With 1H-Benzimidazol-2-Yl(4-((3-(Tetrahydro-2H-Pyran-4-Yl)-2-Pyridinyl)Oxy)Phenyl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-08-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, 2W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: ZN, SO4, 2W1
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Human Gkrp Bound To Amg-0771 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TF, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TF, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-2668
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TG, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TG, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3227 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TJ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TJ, S6P, IOD, GOL, SO4
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Gkrp Bound To Amg0556 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UW, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UW, S6P, IOD, GOL, SO4
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Gkrp Bound To Amg-0471 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5112 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UY, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg5106 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-23 Classification: CARBOHYDRATE BINDING PROTEIN Ligands: 2TO, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 2TO, S6P, IOD, GOL, SO4
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Crystal Structure Of Pde10A With Imidazo[4,5-B]Pyridines As Potent And Selective Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INBHITOR Ligands: ZN, SO4, GOL, 2KR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: ZN, SO4, GOL, 2KR
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Human Gkrp Complexed To Amg-3969 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG9, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG9, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5980 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG0, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG0, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-6861 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-03-12 Classification: SUGAR BINDING PROTEIN Ligands: 2EU, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-12
Ligands: 2EU, S6P, IOD, GOL, SO4
