Search Count: 25
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Crystal Structure Of Kras G12D In Complex With Gdp And Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2023-11-08 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, VM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GDP, MG, VM9
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Crystal Structure Of Kras G12D In Complex With Gdp And Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-11-08 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, VQT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GDP, MG, VQT
 |
Crystal Structure Of Kras G12D In Complex With Gdp And Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2023-11-08 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, VR5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GDP, MG, VR5
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, F4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F4G
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.36 Å Release Date: 2018-05-09 Classification: Transferase/Transferase Inhibitor Ligands: ZN, F4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F4A
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Co-Crystal Structure Of Mnk2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, ET8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, ET8
 |
Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.38 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, FYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, FYV
 |
Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, F4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F4J
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Co-Crytsal Structure Of Mnk2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, F67, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F67, CL
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.32 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, N45 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, N45
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Co-Crystal Structure Of Mnk2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, FZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, FZJ
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The Novel P300/Cbp Inhibitor A-485 Uncovers A Unique Mechanism Of Action To Target Ar In Castrate Resistant Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-09-27 Classification: transferase/transferase INHIBITOR Ligands: 6TF, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: 6TF, NA
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Crystal Structure Of Human Nampt With A-1293201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: 7T7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7T7, SO4
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Crystal Structure Of Human Nampt With A-1326133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 7TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: SO4, 7TA
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HY
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HV
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Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(2-Methoxyphenyl)Methyl]-N,N-Dimethyl-4-(1-Methylindol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING, INHIBITOR Ligands: LQD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: LQD
 |
Polycomb Protein Eed In Complex With Inhibitor: 2-[4-(4-{(3S,4R)-4-(Dimethylamino)-1-[(2-Fluoro-6-Methylphenyl)Methyl]Pyrrolidin-3-Yl}Phenyl)-1H-Pyrazol-1-Yl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING, INHIBITOR Ligands: 7XG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 7XG
 |
Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(2-Bromo-6-Fluorophenyl)Methyl]-N,N-Dimethyl-4-(1-Methyl-1H-Indol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: 82D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 82D
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Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(1S)-7-Fluoro-2,3-Dihydro-1H-Inden-1-Yl]-N,N-Dimethyl-4-(1-Methyl-1H-Indol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: 82G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 82G