Search Count: 11
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Structure-Based Design Of Ask1 Inhibitors As Potential First-In-Class Agents For Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 8GV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: SO4, 8GV
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Structure-Based Design Of Ask1 Inhibitors As Potential First-In-Class Agents For Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8GY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 8GY
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Structure-Based Design Of Ask1 Inhibitors As Potential First-In-Class Agents For Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8GS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 8GS
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Human Glucokinase In Complex With Novel Indazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2017-05-31 Classification: transferase/transferase activator Ligands: GLC, 8WM, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: GLC, 8WM, IOD
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Human Glucokinase In Complex With Novel Pyrazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2017-05-31 Classification: transferase/transferase activator Ligands: GLC, 8WJ, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: GLC, 8WJ, IOD
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Potent, Reversible Metap2 Inhibitors Via Fragment Based Drug Discovery
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-05-25 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MN, DMS, EDO, 6KP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, DMS, EDO, 6KP
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Potent, Reversible Metap2 Inhibitors Via Fbdd
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-05-25 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MN, GOL, DMS, 6KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, GOL, DMS, 6KO
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Potent, Reversible Metap2 Inhibitors Via Fbdd
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-05-25 Classification: Hydrolase4/Hydrolase Inhibitor Ligands: MN, SO4, 6KN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, SO4, 6KN
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Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-(6-Fluoro-4-Oxoquinazolin-3(4H)-Yl)-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 1FW, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: GLC, 1FW, IOD
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Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-(6-Fluoro-2,4-Dioxo-1,4-Dihydroquinazolin-3(2H)-Yl)-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 1FX, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: GLC, 1FX, IOD
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Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-[4-(Methylsulfonyl)-2-Oxopiperazin-1-Yl]-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 1FY, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: GLC, 1FY, IOD