Search Count: 20
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(((3R,4R,5S)-3-((4,4-Difluorocyclohexyl)Methoxy)-5-Methoxypiperidin-4-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XX, SO4
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N-Terminal Bromodomain Of Human Brd4 With 8-(((3R,4R,5S)-3-((4,4-Difluorocyclohexyl)Methoxy)-5-Methoxypiperidin-4-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XX
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N-Terminal Bromodomain Of Human Brd4 With 5-(5-Aminopyridin-3-Yl)-8-(((3R,4R)-3-((1,1-Dioxidotetrahydro-2H-Thiopyran-4-Yl)Methoxy)Piperidin-4-Yl)Amino)-3-Methyl-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XW
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Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-2-(4- Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: N1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: N1D
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Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1- Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: TVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: TVU
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Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, XZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, XZB
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Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Ethyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, H1B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, H1B
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N-Terminal Bromodomain Of Human Brd4 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2- Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: CA, EDO, TVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: CA, EDO, TVU
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N-Terminal Bromodomain Of Human Brd4 With N-(1,1-Dioxo-1-Thian-4-Yl)- 5-Methyl-4-Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C- Pyridine-2-Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, 5V2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, 5V2
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N-Terminal Bromodomain Of Human Brd4 With 7-(3,4-Dimethoxyphenyl)-2-(4-Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, N1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, N1D
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Jmjd2A Complexed With 8-Hydroxyquinoline-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2014-02-05 Classification: OXIDOREDUCTASE Ligands: NI, ZN, CL, 8HQ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-05
Ligands: NI, ZN, CL, 8HQ, GOL
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Crystal Structure Of Alkb In Complex With 5-Carboxy-8-Hydroxyquinoline (Iox1)
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2013-06-26 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: 8XQ, MN, ACT, DMS |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: 8XQ, MN, ACT, DMS
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Factor Inhibiting Hif-1 Alpha In Complex With 8-Hydroxyquinoline-5- Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-04-24 Classification: OXIDOREDUCTASE Ligands: FE, 8XQ, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: FE, 8XQ, SO4, GOL
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Factor Inhibiting Hif-1 Alpha In Complex With Daminozide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-10-03 Classification: OXIDOREDUCTASE Ligands: SO4, GOL, DZA, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: SO4, GOL, DZA, ZN
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Jmjd2A Complexed With Daminozide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2012-10-03 Classification: OXIDOREDUCTASE Ligands: NI, ZN, CL, DZA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: NI, ZN, CL, DZA, GOL
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Histone Lysine Demethylase Jmjd2A In Complex With T11C Peptide Substrate Crosslinked To N-Oxalyl-D-Cysteine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-02-08 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE SUBSTRATE Ligands: NI, ZN, 08P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: NI, ZN, 08P
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Crystal Structure Of The Coiled Coil Domain Of Beclin 1, An Essential Autophagy Protein
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-01-18 Classification: APOPTOSIS |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
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Structure Of Human Phosphorylase Kinase, Gamma 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-02-09 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: B49
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Crystal Structure Of The Middle Domain Of Human Hsp90-Beta Refined At 2.3 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2010-12-15 Classification: CHAPERONE Ligands: SO4, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: SO4, GOL, EDO
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Crystal Structure Of The Human Jmjd3 Jumonji Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-11-24 Classification: OXIDOREDUCTASE Ligands: NI, NA, EDO, 8XQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-24
Ligands: NI, NA, EDO, 8XQ