Search Count: 19
![]() |
Crystal Structure Of Inhibitor Gne-6893 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2024-10-02 Classification: SIGNALING PROTEIN Ligands: A1APL, DMS, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1APL, DMS, NA
![]() |
Crystal Structure Of Inhibitor 1 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2024-10-02 Classification: SIGNALING PROTEIN Ligands: EDO, A1APO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: EDO, A1APO
![]() |
Crystal Structure Of Inhibitor Gne-6893 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2024-10-02 Classification: SIGNALING PROTEIN Ligands: MES, EDO, DMS, A1APR, NA, PEG, A1APQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: MES, EDO, DMS, A1APR, NA, PEG, A1APQ
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2YE
![]() |
Crystal Structure Of Hpk1 In Complex With Gne1858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F97, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: F97, EDO, MES
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2WI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2WI, SO4
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2TR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2TR
![]() |
Structure Of The Vps34 Kinase Domain With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-11-24 Classification: TRANSFERASE/TRANSFERASE inhibitor |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
![]() |
Structure Of The Vps34 Kinase Domain With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2021-11-24 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: GOL, 7IK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: GOL, 7IK
![]() |
Structure Of The Vps34 Kinase Domain With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-11-24 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7IQ, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: 7IQ, GOL, NA
![]() |
Pim1 In Complex With Cpd16 (5-Amino-N-(5-((4R,5R)-4-Amino-5-Fluoroazepan-1-Yl)-1-Methyl-1H-Pyrazol-4-Yl)-2-(2,6-Difluorophenyl)Thiazole-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: GOL, PO4, KUV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: GOL, PO4, KUV
![]() |
Co-Crystal Structure Of Dengue Virus Serotype 2 Rna Dependent Rna Polymerase With Compound 27
Organism: Dengue virus 2
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2016-08-24 Classification: HYDROLASE Ligands: ZN, 68T, MES |
Organism: Dengue virus 2
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: ZN, 68T, MES
![]() |
Dengue Serotype 3 Rna-Dependent Rna Polymerase Bound To Compound 27
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 68T |
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, 68T
![]() |
Dengue Serotype 3 Rna-Dependent Rna Polymerase Bound To Compound 29
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 68E |
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, 68E
![]() |
Dengue 3 Ns5 Protein With Compound 29
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, SAH, 68E, EDO, MG, PEG |
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, SAH, 68E, EDO, MG, PEG
![]() |
Dengue 3 Ns5 Protein With Compound 27
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, PEG, 6L2, MG, EDO, SAH |
Organism: Dengue virus 3
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, PEG, 6L2, MG, EDO, SAH
![]() |
Discovery Of 3,5-Substituted 6-Azaindazoles As Potent Pan-Pim Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-10-28 Classification: Transferase/Transferase Inhibitor Ligands: L20, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: L20, PO4
![]() |
Pim1 In Complex With Cpd4 (3-Methyl-5-(Pyridin-3-Yl)-1H-Pyrazolo[3,4-C]Pyridine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2015-10-28 Classification: Transferase/Transferase Inhibitor Ligands: 5E5, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 5E5, PO4
![]() |
Pim1 In Complex With Cpd36 ((1S,3S)-N1-(6-(5-(Pyridin-3-Yl)-1H-Pyrazolo[3,4-C]Pyridin-3-Yl)Pyridin-2-Yl)Cyclohexane-1,3-Diamine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2015-10-28 Classification: Transferase/Transferase Inhibitor Ligands: 5E6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 5E6
