Search Count: 23
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Crystal Structure Of Jak1 In Complex With Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2016-11-09 Classification: TRANSFERASE Ligands: ADP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: ADP, MG
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Crystal Structure Of Jak1 In Complex With Pf-4950736
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-11-09 Classification: transferase/transferase INHIBITOR Ligands: 6TE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6TE
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Ampk Bound To Allosteric Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.41 Å Release Date: 2016-08-17 Classification: TRANSFERASE Ligands: STU, 6VT, CL, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: STU, 6VT, CL, AMP, ADP, SO4
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Structure Of Ampk In Complex With Staurosporine Inhibitor And In The Absence Of A Synthetic Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.46 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor Ligands: STU, CL, SO4, AMP |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, CL, SO4, AMP
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Structure Of Ampk In Complex With Cl-A769662 Activator And Staurosporine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor/activator Ligands: STU, CL, 32J, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, CL, 32J, AMP, ADP, SO4
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Structure Of Ampk In Complex With Br2-A769662Core Activator And Staurosporine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.55 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor/activator Ligands: STU, 32H, CL, AMP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, 32H, CL, AMP, SO4
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Crystal Structure Of Itk In Complex With Compound 1 [4-(Carbamoylamino)-1-(Naphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Y
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Crystal Structure Of Itk In Complex With Compound 5 {4-(Carbamoylamino)-1-(7-Methoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide}
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Z
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Crystal Structure Of Itk In Complex With Compound 7 [4-(Carbamoylamino)-1-(7-Ethoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1YZ
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Crystal Structure Of Itk In Complex With Compound 8 [4-(Carbamoylamino)-1-(7-Propoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1E0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1E0
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide] And Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS, ADP
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Cdk-2 With Indazole Inhibitor 17 Bound At Its Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-02-03 Classification: TRANSFERASE/Transferase inhibitor Ligands: EZR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-03
Ligands: EZR
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Cdk-2 With Indazole Inhibitor 9 Bound At Its Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2009-02-03 Classification: TRANSFERASE Ligands: EZV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-03
Ligands: EZV
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Cdk-2-Cyclin Complex With Indazole Inhibitor 9 Bound At Its Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-02-03 Classification: Transferase/Cell cycle Ligands: GOL, EZV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-03
Ligands: GOL, EZV, SO4
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Thermodynamic And Structure Guided Design Of Statin Hmg-Coa Reductase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: 3HI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: 3HI
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Thermodynamic And Structure Guided Design Of Statin Hmg-Coa Reductase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: 4HI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: 4HI
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Thermodynamic And Structure Guided Design Of Statin Hmg-Coa Reductase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: SO4, 5HI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: SO4, 5HI
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Thermodynamic And Structure Guided Design Of Statin Hmg-Coa Reductase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: 6HI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: 6HI
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Thermodynamic And Structure Guided Design Of Statin Hmg-Coa Reductase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: SO4, 7HI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: SO4, 7HI
