Search Count: 55
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Crystal Structure Of Mouse Btk Kinase Domain In Complex With Compound 9A
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: JVP |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: JVP
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Human Retenoid-Related Orphan Receptor-Gamma Ligand- Binding Domain In Complex With Indole Ligand Cp9B In Inverse Agonist Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN Ligands: F7M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: F7M
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Rorc2 Lbd Complexed With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN Ligands: F7J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: F7J
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Crystal Structure Of Jak1 In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2018-01-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: D7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D7D
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Crystal Structure Of Jak2 In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-01-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: D7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D7D
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Crystal Structure Of Jak1 In Complex With Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2016-11-09 Classification: TRANSFERASE Ligands: ADP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: ADP, MG
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Crystal Structure Of Jak1 In Complex With Pf-4950736
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-11-09 Classification: transferase/transferase INHIBITOR Ligands: 6TE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6TE
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Ampk Bound To Allosteric Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.41 Å Release Date: 2016-08-17 Classification: TRANSFERASE Ligands: STU, 6VT, CL, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: STU, 6VT, CL, AMP, ADP, SO4
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Structure Of Ampk In Complex With Staurosporine Inhibitor And In The Absence Of A Synthetic Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.46 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor Ligands: STU, CL, SO4, AMP |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, CL, SO4, AMP
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Structure Of Ampk In Complex With Cl-A769662 Activator And Staurosporine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor/activator Ligands: STU, CL, 32J, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, CL, 32J, AMP, ADP, SO4
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Structure Of Ampk In Complex With Br2-A769662Core Activator And Staurosporine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.55 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor/activator Ligands: STU, 32H, CL, AMP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, 32H, CL, AMP, SO4
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Crystal Structure Of Pbp3 In Complex With Compound 14 ((2E)-2-({[(2S)-2-{[(2Z)-2-(2-Amino-1,3-Thiazol-4-Yl)-2-{[(1,5-Dihydroxy-4-Oxo-1,4-Dihydropyridin-2-Yl)Methoxy]Imino}Acetyl]Amino}-3-Oxopropyl]Oxy}Imino)Pentanedioic Acid)
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-05-07 Classification: transferase/transferase inhibitor Ligands: 2U2 |
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: 2U2
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Crystal Structure Of Pbp3 In Complex With Bal30072 ((2Z)-2-(2-Amino-1,3-Thiazol-4-Yl)-2-{[(1,5-Dihydroxy-4-Oxo-1,4-Dihydropyridin-2-Yl)Methoxy]Imino}-N-{(2S)-1-Hydroxy-3-Methyl-3-[(Sulfooxy)Amino]Butan-2-Yl}Ethanamide)
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-05-07 Classification: transferase/transferase inhibitor Ligands: 2U3 |
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: 2U3
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Crystal Structure Of Pbp1A In Complex With Compound 17 ((4Z,8S,11E,14S)-5-(2-Amino-1,3-Thiazol-4-Yl)-14-(5,6-Dihydroxy-1,3-Dioxo-1,3-Dihydro-2H-Isoindol-2-Yl)-8-Formyl-2-Methyl-6-Oxo-3,10-Dioxa-4,7,11-Triazatetradeca-4,11-Diene-2,12,14-Tricarboxylic Acid)
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2014-05-07 Classification: transferase/transferase inhibitor Ligands: 2U4 |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: 2U4
 |
Crystal Structure Of Itk In Complex With Compound 1 [4-(Carbamoylamino)-1-(Naphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Y
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Crystal Structure Of Itk In Complex With Compound 5 {4-(Carbamoylamino)-1-(7-Methoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide}
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Z
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Crystal Structure Of Itk In Complex With Compound 7 [4-(Carbamoylamino)-1-(7-Ethoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1YZ
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Crystal Structure Of Itk In Complex With Compound 8 [4-(Carbamoylamino)-1-(7-Propoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1E0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1E0
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide] And Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS, ADP