Search Count: 12
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Ternary Complex Structure Of Compound 1 Bound To Smarca2 Bromodomain And Dcaf16:Ddb1Deltabpb
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-05-20 Classification: TRANSCRIPTION Ligands: ZN, A1JLV |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-05-20
Ligands: ZN, A1JLV
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Pvhl:Elob:Eloc In Complex With (2S,4R)-1-((S)-2-(1-Fluorocyclopropane-1-Carboxamido)-3,3-Dimethylbutanoyl)-4-Hydroxy-N-((S)-1-(2-Methyl-4-(4-Methylthiazol-5-Yl)Phenyl)Ethyl)Pyrrolidine-2-Carboxamide (Compound 37)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2023-09-27 Classification: LIGASE Ligands: VFO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-27
Ligands: VFO
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Pvhl:Elob:Eloc In Complex With (2S,4R)-1-((S)-2-(1-Fluorocyclopropane-1-Carboxamido)-3,3-Dimethylbutanoyl)-4-Hydroxy-N-((S)-1-(2-Methyl-4-(4-Methylthiazol-5-Yl)Phenyl)Ethyl)Pyrrolidine-2-Carboxamide (Compound 30)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2023-09-27 Classification: LIGASE Ligands: VYQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-27
Ligands: VYQ
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Pvhl:Elob:Eloc In Complex With (2S,4R)-N-((S)-1-(5-Fluoro-2-Methoxy-4-(4-Methylthiazol-5-Yl)Phenyl)Ethyl)-1-((S)-2-(1-Fluorocyclopropane-1-Carboxamido)-3,3-Dimethylbutanoyl)-4-Hydroxypyrrolidine-2-Carboxamide (Compound 33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2023-09-27 Classification: LIGASE Ligands: VH3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-27
Ligands: VH3
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Ternary Structure Of Intramolecular Bivalent Glue Degrader Ibg1 Bound To Brd4 And Dcaf16:Ddb1Deltabpb
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-05-17 Classification: TRANSCRIPTION Ligands: ZN, U79 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-05-17
Ligands: ZN, U79
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Crystal Structure Of Socs2:Elonginb:Elonginc In Complex With Compound Mn551
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2023-04-26 Classification: LIGASE Ligands: JIH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: JIH
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Crystal Structure Of Socs2:Elonginb:Elonginc In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-04-26 Classification: LIGASE Ligands: JI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: JI9
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Crystal Structure Of Socs2:Elonginb:Elonginc In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2023-04-26 Classification: LIGASE Ligands: JI0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: JI0
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Crystal Structure Of Socs2:Elonginb:Elonginc In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2023-04-26 Classification: LIGASE Ligands: JHR, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: JHR, PO4
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Crystal Structure Of Socs2:Elonginb:Elonginc In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2023-04-26 Classification: LIGASE Ligands: JH9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: JH9
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Co-Crystal Structure Of Socs2:Elonginb:Elonginc In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2023-04-26 Classification: LIGASE Ligands: EDO, JH9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: EDO, JH9
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Crystal Structure Of At7 In Complex With The Second Bromodomain Of Human Brd4 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IZR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IZR
