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Search Count: 19

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7EI2 image
Structure Of Human Nnmt In Complex With Macrocyclic Peptide 8

7EGU image
Structure Of Human Nnmt In Complex With Macrocyclic Peptide X

7EHZ image
Structure Of Human Nnmt In Complex With Macrocyclic Peptide 2

6N3L image
Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents

6N3N image
Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents

6N3O image
Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents

5U4X image
Coactivator-Associated Arginine Methyltransferase 1 With Tp-064
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.88 Å Release Date: 2016-12-21
Classification: TRANSFERASE
Ligands: SAH, 7VM, UNX

3W2O image
Egfr Kinase Domain T790M/L858R Mutant With Tak-285

3W2P image
Egfr Kinase Domain T790M/L858R Mutant With Compound 2

3W2Q image
Egfr Kinase Domain T790M/L858R Mutant With Hki-272

3W2R image
Egfr Kinase Domain T790M/L858R Mutant With Compound 4

3W2S image
Egfr Kinase Domain With Compound4

2ZJH image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-(1-Benzyl-Piperidin-4-Yl)-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1H

2ZJI image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(2,6-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1I

2ZJJ image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid (2-Mercapto-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1J

2ZJK image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid(3-Mercapto-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1K

2ZJL image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Bromo-2,3-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1L

2ZJM image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Chloro-2-Isopropoxy-3-Methoxy-Benzyl)-Piperidin-4-Yl]-2-(4-Sulfamoyl-Phenoxy)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1M

2ZJN image
Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Chloro-2-Isopropoxy-3-Methoxy-Benzyl)-Piperidin-4-Yl]-2-(2-Methyl-4-Sulfamoyl-Phenoxy)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2009-01-20
Classification: HYDROLASE
Ligands: F1N
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