Search Count: 12
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Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
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Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
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Selective Small Molecule Inhibition Of The Fmn Riboswitch
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2015-10-07 Classification: RNA/INHIBITOR Ligands: K, MG, 51B |
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: K, MG, 51B
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Discovery Of Novel, Dual Mechanism Erk Inhibitors By Affinity Selection Screening Of An Inactive Kinase State
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-11-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3G7, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: 3G7, SO4
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Ternary Complex With Compound 1, Atp-Gs And Mg2P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: 3BM, AGS, MG, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: 3BM, AGS, MG, CA, NA
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Binary Complex With Atp-Gs And Mg2P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: AGS, MG, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: AGS, MG, CA, NA
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Binary Complex With K252A And Mg2P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: KSA, MG, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: KSA, MG, CA, NA
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Ternary Complex With Pd, Adp And Mg2P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: ADP, MG, CA, NA, 4BM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: ADP, MG, CA, NA, 4BM
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Ternary Complex With U0126, Adp And Mg2P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: 5BM, ADP, MG, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: 5BM, ADP, MG, CA, NA
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Binary Complex With Adp And Mg2P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: ADP, MG, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: ADP, MG, CA, NA
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Docking And Dimerization Domain (D/D) Of The Type Ii-Alpha Regulatory Subunity Of Protein Kinase A (Pka) In Complex With A Peptide From An A-Kinase Anchoring Protein
Organism: Rattus norvegicus
Method: SOLUTION NMR Release Date: 2006-08-29 Classification: TRANSFERASE |
Organism: Rattus norvegicus
Method: SOLUTION NMR
Release Date: 2006-08-29
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Docking And Dimerization Domain (D/D) Of The Regulatory Subunit Of The Type Ii-Alpha Camp-Dependent Protein Kinase A Associated With A Peptide Derived From An A-Kinase Anchoring Protein (Akap)
Organism: Rattus norvegicus
Method: SOLUTION NMR Release Date: 2006-08-29 Classification: TRANSFERASE |
Organism: Rattus norvegicus
Method: SOLUTION NMR
Release Date: 2006-08-29