Search Count: 18
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G-925 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2022-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GGU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: GGU
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G-059 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2022-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GJN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: GJN
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.13 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: QRY, CL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: QRY, CL, SO4
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Crystal Structure Of The P300 Acetyltransferase Domain With Peptide-Competitive Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, QS4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: COA, QS4, DMS
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: SO4, CL, QS1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: SO4, CL, QS1
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: QSD, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: QSD, SO4, CL
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Structure Of Human Polycomb Repressive Complex 2 (Prc2) With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.47 Å Release Date: 2017-02-22 Classification: Transferase/Inhibitor Ligands: ZN, 74D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 74D
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Structure Of G9A Set-Domain With Histone H3K9Norleucine Mutant Peptide And Bound S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: ZN, SAM
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Structure Of G9A Set-Domain With Histone H3K9Ala Mutant Peptide And Bound S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2016-07-06 Classification: TRANSFERASE Ligands: ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, SAM
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Structure Of G9A Set-Domain With Histone H3K9M Mutant Peptide And Bound S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-07-06 Classification: TRANSFERASE Ligands: ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, SAM
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Structure Of G9A Set-Domain With Histone H3K9M Peptide And Excess Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-07-06 Classification: TRANSFERASE Ligands: ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: ZN, SAM
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02773986
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: SCN, 68Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: SCN, 68Y
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02778174
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: EDO, SCN, 69A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: EDO, SCN, 69A
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02857790
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: ACT, CA, 69B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ACT, CA, 69B
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Cbp In Complex With Cpd23 ((R)-6-(3-(Benzyloxy)Phenyl)-4-Methyl-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69F, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69F, B3P, EDO, NA, PEG
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Cbp In Complex With Cpd637 ((R)-4-Methyl-6-(1-Methyl-3-(1-Methyl-1H-Pyrazol-4-Yl)-1H-Indazol-5-Yl)-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69E, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69E, B3P, EDO, NA, PEG
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Cpi-0610
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2016-02-10 Classification: TRANSCRIPTION Ligands: 62G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 62G
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Benzoisoxazoloazepine 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-02-10 Classification: TRANSCRIPTION Ligands: 62V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 62V