Search Count: 27
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Crystal Structure Of Human Kras G12C Covalently Bound To Amg 510
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-11-06 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: MG, GDP, MOV
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Hmcl1 Inhibitor Complex
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2019-05-22 Classification: APOPTOSIS/INHIBITOR Ligands: N8J |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2019-05-22
Ligands: N8J
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Co-Crystal Structure Of Mcl1 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-05-15 Classification: APOPTOSIS/INHIBITOR Ligands: LOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: LOD
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Co-Crystal Structure Of Mcl1 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-05-15 Classification: APOPTOSIS/INHIBITOR Ligands: LOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: LOJ
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Co-Crystal Structure Of Mcl1 With Inhibitor 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-05-15 Classification: APOPTOSIS/INHIBITOR Ligands: N0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: N0J
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Crystal Structure Of Mcl1 With Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2019-05-15 Classification: APOPTOSIS/INHIBITOR Ligands: N0M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: N0M
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Crystal Structure Of Mcl1 With Inhibitor 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-05-15 Classification: APOPTOSIS Ligands: N0P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: N0P
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Co-Crystal Structure Of Mdm2 In Complex With Am-7209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2014-12-03 Classification: LIGASE/LIGASE INHIBITOR Ligands: 3UD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: 3UD, SO4
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Co-Crystal Structure Of Mdm2 (17-111) With Compound 16, {(3R,5R,6S)-5-(3-Chlorophenyl)-6-(4-Chlorophenyl)-1-[(1S)-1-(6-Cyclopropylpyridin-2-Yl)Propyl]-3-Methyl-2-Oxopiperidin-3-Yl}Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-07-16 Classification: Ligase/Ligase inhibitor Ligands: 35S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: 35S
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Co-Crystal Structure Of Mdm2(17-111) In Complex With Compound 48
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-04-02 Classification: ligase/ligase inhibitor Ligands: 2TZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2TZ
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U0, SO4
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 47
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U1
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Co-Crystal Structure Of Mdm2 With Inhbitor Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U5, SO4
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Co-Crystal Structure Of Mdm2 With Inhbitor Compound 46
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U6, SO4
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U7
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-03-19 Classification: ligase/ligase inhibitor Ligands: 2TW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: 2TW
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Co-Crystal Structure Of Mdm2 (17-111) In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-02-19 Classification: ligase/ligase inhibitor Ligands: 2SW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-19
Ligands: 2SW, SO4
