Search Count: 62
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X-Ray Structure Of Furin Bound To Bos-318, A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2022-01-12 Classification: HYDROLASE/INHIBITOR Ligands: CA, XTA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: CA, XTA, EDO
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Crystal Structure Of Matriptase1 In Complex With A Peptidomimetic Benzothiazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2019-10-02 Classification: hydrolase/hydrolase inhibitor Ligands: MG, EOH, GSH, KD7, 144 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-02
Ligands: MG, EOH, GSH, KD7, 144
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X-Ray Structure Of Polypeptide Deformylase
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-06-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, NB4 |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: NI, NB4
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X-Ray Structure Of Polypeptide Deformylase With A Piperazic Acid
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2019-06-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, SO4, N9Y |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: NI, SO4, N9Y
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Crystal Structure Of Rip1 Kinase In Complex With A Pyrrolidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2019-05-08 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: M5J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: M5J, SO4
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Crystal Structure Of Rip1 Kinase In Complex With Dhp77
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: JSW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: JSW
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C-Abl Kinase Domain With The Activator(Cmpd6), 2-Cyano-N-(4-(3,4-Dichlorophenyl)Thiazol-2-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-03-13 Classification: TRANSFERASE Ligands: SO4, STI, KWD, 2PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: SO4, STI, KWD, 2PE
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C-Abl Kinase Domain With The Activator(Cmpd29), N-(1-(3,4-Dichlorophenyl)-4,5-Dihydro-1H-Pyrazol-3-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-03-13 Classification: TRANSFERASE Ligands: STI, KWV, SO4, GOL, 2PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: STI, KWV, SO4, GOL, 2PE
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C-Abl Kinase Domain With The Activator(Cmpd51), N-(1-(3,4-Dichlorophenyl)-4-(2-Hydroxyethyl)-4,5-Dihydro-1H-Pyrazol-3-Yl)Isonicotinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2019-03-13 Classification: TRANSFERASE Ligands: SO4, STI, KWP, GOL, 2PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: SO4, STI, KWP, GOL, 2PE
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Rip1 Kinase ( Flag 1-294, C34A, C127A, C233A, C240A) With Gsk772
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-07-05 Classification: transferase/transferase inhibitor Ligands: 7MJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: 7MJ
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Crystal Structure Of Unglycosylated Apo Human Furin @1.89A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-05-04 Classification: HYDROLASE Ligands: CA, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: CA, PO4, EDO
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Crystal Structure Of Human Hexokinase 2 With Cmpd 30, A 2-Amino-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 604 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 604
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Crystal Structure Of Human Hexokinase 2 With Cmpd 27, A 2-Amido-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 603 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 603
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Crystal Structure Of Human Hexokinase 2 With Cmpd 1, A C-2-Substituted Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 62C, BG6, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 62C, BG6, FLC
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Crystal Structure Of Rip1 Kinase With A Benzo[B][1,4]Oxazepin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 65U
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Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With A Type Iii Kinase Inhibitor (Gsk2850163A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2015-11-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4K7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 4K7
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Crystal Structure Of Pire1Alpha In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2015-11-11 Classification: Transferase/transferase inhibitor Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: STU