Search Count: 47
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Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION Ligands: Q0S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q0S
 |
Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION Ligands: Q0M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q0M
 |
Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION/INHIBITOR Ligands: Q0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q0Y
 |
Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION Ligands: Q1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q1J
 |
Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION Ligands: Q1M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q1M
 |
Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION Ligands: Q1P, Q1S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q1P, Q1S
 |
Discovery And Optimization Of Salicyclic Acid-Derived Sulfonamide Inhibitors Of The Wdr5:Myc Protein-Protein Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-04 Classification: TRANSCRIPTION Ligands: Q1G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q1G
 |
Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2018-09-05 Classification: dna binding protein/inhibitor |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
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Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2018-09-05 Classification: dna binding protein/inhibitor Ligands: DMS, G2V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: DMS, G2V
 |
Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-09-05 Classification: dna binding protein/inhibitor Ligands: G1Y, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: G1Y, DMS
 |
Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2018-09-05 Classification: dna binding protein/inhibitor Ligands: G2J, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: G2J, SO4, DMS
 |
Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-07-18 Classification: dna binding protein/inhibitor Ligands: G2D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: G2D
 |
Ligand-Bound Ras:Sos:Ras Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: MG, GNP, 5UU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: MG, GNP, 5UU
 |
Ligand-Bound Ras:Sos:Ras Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: MG, GNP, 5UX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: MG, GNP, 5UX
 |
Ligand-Bound Ras:Sos:Ras Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: MG, GNP, 5UV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: MG, GNP, 5UV
 |
Ligand-Bound Ras:Sos:Ras Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: MG, GNP, 5UW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: MG, GNP, 5UW
 |
Mcl-1 Complexed With Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2018-01-31 Classification: APOPTOSIS Ligands: ECY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-31
Ligands: ECY
 |
Mcl-1 Complexed With Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-01-31 Classification: APOPTOSIS Ligands: ECM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-31
Ligands: ECM
 |
Discovery Of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors Using Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-01-18 Classification: apoptosis/apoptosis inhibitor Ligands: 6AL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 6AL
 |
Discovery Of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors Using Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2017-01-18 Classification: apoptosis/apoptosis inhibitor Ligands: 6AK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 6AK