Search Count: 8
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Crystal Structure Of Brd9 Bromodomain In Complex With Compound Ea-89
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2022-08-10 Classification: TRANSCRIPTION Ligands: L8L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: L8L
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Crystal Structure Of Dot1L In Complex With An Inhibitor (Compound 3).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-12-11 Classification: TRANSFERASE Ligands: N4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: N4W
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Crystal Structure Of Dot1L In Complex With An Inhibitor (Compound 10).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2019-12-11 Classification: TRANSFERASE Ligands: N4Z, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: N4Z, K
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Crystal Structure Of Dot1L In Complex With An Inhibitor (Compound 11).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2019-12-11 Classification: TRANSFERASE Ligands: N5K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: N5K, SO4
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Crystal Structure Of Dot1L In Complex With Inhibitor Cpd2 [2-(2-(5-((2-Chlorophenoxy)Methyl)-1H-Tetrazol-1-Yl)Acetyl)-N-(4-Chlorophenyl)Hydrazinecarboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2016-06-15 Classification: TRANSFERASE Ligands: 5EG, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-15
Ligands: 5EG, K
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Crystal Structure Of Dot1L In Complex With Inhibitor Cpd3 [N-(1-(2-Chlorophenyl)-1H-Indol-6-Yl)-2-(2-(5-(2-Chlorophenyl)-1H-Tetrazol-1-Yl)Acetyl)Hydrazinecarboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2016-06-15 Classification: TRANSFERASE Ligands: K, 5EK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-15
Ligands: K, 5EK
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Crystal Structure Of Dot1L In Complex With Inhibitor Cpd10 [6'-Chloro-1,4-Dimethyl-5'-(2-Methyl-6-((4-(Methylamino)Pyrimidin-2-Yl)Amino)-1H-Indol-1-Yl)-[3,3'-Bipyridin]-2(1H)-One]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2016-06-15 Classification: TRANSFERASE Ligands: K, 5EW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-15
Ligands: K, 5EW
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Crystal Structure Of Dot1L In Complex With Inhibitor Cpd11 [N4-Methyl-N2-(2-Methyl-1-(2-Phenoxyphenyl)-1H-Indol-6-Yl)Pyrimidine-2,4-Diamine]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-06-15 Classification: TRANSFERASE Ligands: 5EV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-15
Ligands: 5EV, SO4
