Search Count: 12
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Crystal Structure Of Trim25 Pryspry Covalently Bound To 2-Chloro-1-[4-(3-Methyl-4-Phenyl-Phenyl)Carbonyl-1,4-Diazepan-1-Yl]Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-05-21 Classification: LIGASE Ligands: A1IZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: A1IZK
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Ligand Zz001229A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2024-02-07 Classification: GENE REGULATION Ligands: EDO, IX4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: EDO, IX4
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Crystal Structure Of The First Bromodomain Of Human Brd4 L94C Variant In Complex With Racemic 3,5-Dimethylisoxazol Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2023-08-02 Classification: GENE REGULATION Ligands: E5Q, V0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-02
Ligands: E5Q, V0R
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N-Terminal Bromodomain Of Human Brd4 With Compound 3Ag
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2021-10-06 Classification: TRANSCRIPTION Ligands: 5Z4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 5Z4
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N-Terminal Bromodomain Of Human Brd4 With Compound 3Bg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2021-10-06 Classification: TRANSCRIPTION Ligands: 5YY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 5YY
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N-Terminal Bromodomain Of Human Brd4 With Compound 5Ef
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-10-06 Classification: TRANSCRIPTION Ligands: 5Z1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 5Z1
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N-Terminal Bromodomain Of Human Brd4 With 3-(3-(But-3-Yn-1-Yl)-3H-Diazirin-3-Yl)-N-(3-Methyl-[1,2,4]Triazolo[4,3-A]Pyridin-8-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2020-10-21 Classification: TRANSCRIPTION Ligands: R5W, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: R5W, EDO
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Pi3 Kinase Delta In Complex With Methyl 5-(4-(5-((4-Isopropylpiperazin-1-Yl)Methyl)Oxazol-2-Yl)-1H-Indazol-6-Yl)-2-Methoxynicotinate
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2017-12-27 Classification: TRANSFERASE Ligands: C5Z |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: C5Z
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Pi3 Kinase Delta In Complex With 4-Fluorophenyl 5-(4-(5-((4-Isopropylpiperazin-1-Yl)Methyl)Oxazol-2-Yl)-1H-Indazol-6-Yl)-2-Methoxynicotinate
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-12-20 Classification: TRANSFERASE Ligands: C5W |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: C5W
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Jmjd2A Complexed With 8-Hydroxyquinoline-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2014-02-05 Classification: OXIDOREDUCTASE Ligands: NI, ZN, CL, 8HQ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-05
Ligands: NI, ZN, CL, 8HQ, GOL
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Crystal Structure Of Alkb In Complex With 5-Carboxy-8-Hydroxyquinoline (Iox1)
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2013-06-26 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: 8XQ, MN, ACT, DMS |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: 8XQ, MN, ACT, DMS
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Factor Inhibiting Hif-1 Alpha In Complex With 8-Hydroxyquinoline-5- Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-04-24 Classification: OXIDOREDUCTASE Ligands: FE, 8XQ, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: FE, 8XQ, SO4, GOL
