Search Count: 22
![]() |
Bruton'S Tyrosine Kinase In Complex With Compound 45
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B9
![]() |
Bruton'S Tyrosine Kinase In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0BG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0BG, DMS
![]() |
Bruton'S Tyrosine Kinase In Complex With Compound 65
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B0
![]() |
Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYV
![]() |
Brd4_Bromodomain2 Complex With Pyrrolopyridone Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYV
![]() |
Brd2_Bromodomain2 Complex With Pyrrolopyridone Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYY
![]() |
Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYY
![]() |
Usp7 In Complex With Ligand Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R44, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R44, ACT
![]() |
Usp7 In Complex With Ligand Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R3Y
![]() |
Usp7 In Complex With Ligand Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R4D
![]() |
Usp7 In Complex With Ligand Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R41
![]() |
Usp7 In Complex With Ligand Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R4J, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R4J, ZN
![]() |
Brd2_Bromodomain1 Complex With Inhibitor 744
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-01-29 Classification: SIGNALING PROTEIN Ligands: EDO, HWV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-29
Ligands: EDO, HWV
![]() |
Brd2_Bromodomain2 Complex With Inhibitor 744
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: HWV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: HWV
![]() |
Brutons Tyrosine Kinase In Complex With Compound 50.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-06-12 Classification: transferase/transferase inhibitor Ligands: L9S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: L9S, EDO
![]() |
Crystal Structure Of Human Pi3K-Gamma In Complex With Quinoline-Containing Inhibitor 5G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-06-21 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 6RF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: SO4, 6RF
![]() |
Crystal Structure Of Mouse Aurora A (Asn186->Gly, Lys240->Arg, Met302->Leu) In Complex With 1-(3-Chloro-Phenyl)-3-{5-[2-(Thieno[3,2-D]Pyrimidin-4-Ylamino)- Ethyl]-Thiazol-2-Yl}-Urea [Sns-314]
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-05-12 Classification: TRANSFERASE Ligands: AK2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-05-12
Ligands: AK2
![]() |
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 257
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: 2FR |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: 2FR
![]() |
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 094
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: 3FR |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: 3FR
![]() |
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 557
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:3.32 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: 4FR |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: 4FR
