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7N4Q image
Bruton'S Tyrosine Kinase In Complex With Compound 45
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2022-05-18
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 0B9

7N4R image
Bruton'S Tyrosine Kinase In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.62 Å Release Date: 2022-05-18
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 0BG, DMS

7N4S image
Bruton'S Tyrosine Kinase In Complex With Compound 65
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2022-05-18
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 0B0

6VIW image
Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.43 Å Release Date: 2020-05-06
Classification: SIGNALING PROTEIN
Ligands: QYV

6VIX image
Brd4_Bromodomain2 Complex With Pyrrolopyridone Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.12 Å Release Date: 2020-05-06
Classification: SIGNALING PROTEIN
Ligands: QYV

6VIY image
Brd2_Bromodomain2 Complex With Pyrrolopyridone Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2020-05-06
Classification: SIGNALING PROTEIN
Ligands: QYY

6VIZ image
Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.39 Å Release Date: 2020-05-06
Classification: SIGNALING PROTEIN
Ligands: QYY

6VN2 image
Usp7 In Complex With Ligand Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.93 Å Release Date: 2020-04-29
Classification: HYDROLASE
Ligands: R44, ACT

6VN3 image
Usp7 In Complex With Ligand Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.73 Å Release Date: 2020-04-29
Classification: HYDROLASE
Ligands: R3Y

6VN4 image
Usp7 In Complex With Ligand Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.69 Å Release Date: 2020-04-29
Classification: HYDROLASE
Ligands: R4D

6VN5 image
Usp7 In Complex With Ligand Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2020-04-29
Classification: HYDROLASE
Ligands: R41

6VN6 image
Usp7 In Complex With Ligand Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.99 Å Release Date: 2020-04-29
Classification: HYDROLASE
Ligands: R4J, ZN

6ONY image
Brd2_Bromodomain1 Complex With Inhibitor 744
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.98 Å Release Date: 2020-01-29
Classification: SIGNALING PROTEIN
Ligands: EDO, HWV

6E6J image
Brd2_Bromodomain2 Complex With Inhibitor 744
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.44 Å Release Date: 2019-07-31
Classification: SIGNALING PROTEIN
Ligands: HWV

6NZM image
Brutons Tyrosine Kinase In Complex With Compound 50.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2019-06-12
Classification: transferase/transferase inhibitor
Ligands: L9S, EDO

5KAE image
Crystal Structure Of Human Pi3K-Gamma In Complex With Quinoline-Containing Inhibitor 5G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.65 Å Release Date: 2017-06-21
Classification: Transferase/Transferase Inhibitor
Ligands: SO4, 6RF

3D15 image
Crystal Structure Of Mouse Aurora A (Asn186->Gly, Lys240->Arg, Met302->Leu) In Complex With 1-(3-Chloro-Phenyl)-3-{5-[2-(Thieno[3,2-D]Pyrimidin-4-Ylamino)- Ethyl]-Thiazol-2-Yl}-Urea [Sns-314]
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2009-05-12
Classification: TRANSFERASE
Ligands: AK2

3DBC image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 257
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.35 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 2FR

3DBD image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 094
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.05 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 3FR

3DBE image
Crystal Structure Of An Activated (Thr->Asp) Polo-Like Kinase 1 (Plk1) Catalytic Domain In Complex With Compound 557
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Resolution:3.32 Å Release Date: 2008-10-07
Classification: TRANSFERASE
Ligands: 4FR
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