Search Count: 12
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Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: X3N, ZWE
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Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To H1047R Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERSE INHIBITOR Ligands: EDO, X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: EDO, X3N, ZWE
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Map4K4 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-01-13 Classification: TRANSFERASE/INHIBITOR Ligands: 5DF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: 5DF
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Crystal Structure Of Pyk2 With The Pyrazole 13A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-11-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0YH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: 0YH
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Crystal Structure Of Pyk2 With The Indole 10C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2012-11-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0YJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: 0YJ
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Crystal Structure Of Pyk2 Complexed With Pf-2318841
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-06-23 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 349, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-23
Ligands: 349, PO4
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Crystal Structure Of Pyk2 In Complex With Sulfoximine-Substituted Trifluoromethylpyrimidine Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-05-26 Classification: TRANSFERASE Ligands: SO4, P1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-05-26
Ligands: SO4, P1E
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Crystal Structure Of Pyk2-Apo, Proline-Rich Tyrosine Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-03-31 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-31
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Crystal Structure Of Pyk2 Complexed With Atpgs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-03-31 Classification: TRANSFERASE Ligands: AGS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-31
Ligands: AGS, SO4
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Crystal Structure Of Pyk2 Complexed With Pf-431396
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-03-31 Classification: TRANSFERASE Ligands: 3JZ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-31
Ligands: 3JZ, PO4
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Crystal Structure Of Pyk2 Complexed With Birb796
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2009-03-31 Classification: TRANSFERASE Ligands: B96 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-31
Ligands: B96
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Crystal Structure Of Pyk2 Complexed With Pf-4618433
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-03-31 Classification: TRANSFERASE Ligands: 4JZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-31
Ligands: 4JZ
