Search Count: 26
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Structure Of Ciap1 With Bccov
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-03-08 Classification: APOPTOSIS Ligands: ZN, TO0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, TO0
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Structure Of Ciap1, Btk And Bccov
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2023-03-08 Classification: ONCOPROTEIN Ligands: TOO, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: TOO, ZN
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Crystal Structure Of Jak2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWM
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Structure Of Ciap With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-11-18 Classification: LIGASE Ligands: ZN, TKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: ZN, TKY
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Ternary Complex Structure - Btk Ciap Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-11-18 Classification: LIGASE/TRANSFERASE Ligands: TL7, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: TL7, ZN
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Ternary Complex Structure - Btk Ciap Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.80 Å Release Date: 2020-11-18 Classification: LIGASE/TRANSFERASE Ligands: TKY, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: TKY, ZN
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Tyk2 With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G5D
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Tyk2 With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G4J
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Jak1 With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G4J
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Crystal Structure Of Jak1 In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2018-01-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: D7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D7D
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Crystal Structure Of Jak2 In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-01-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: D7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D7D
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Jak3 With Covalent Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KU
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Jak3 With Covalent Inhibitor 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KV, SO4
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Jak3 With Covalent Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KX
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Jak3 With Covalent Inhibitor Pf-06651600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-11-09 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7H4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 7H4, SO4
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Covalent Inhibitor Of Lyplal1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-07-20 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 6WG, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: 6WG, NO3
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Crystal Structure Of Pbp3 In Complex With Compound 14 ((2E)-2-({[(2S)-2-{[(2Z)-2-(2-Amino-1,3-Thiazol-4-Yl)-2-{[(1,5-Dihydroxy-4-Oxo-1,4-Dihydropyridin-2-Yl)Methoxy]Imino}Acetyl]Amino}-3-Oxopropyl]Oxy}Imino)Pentanedioic Acid)
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-05-07 Classification: transferase/transferase inhibitor Ligands: 2U2 |
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: 2U2
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Crystal Structure Of Pbp3 In Complex With Bal30072 ((2Z)-2-(2-Amino-1,3-Thiazol-4-Yl)-2-{[(1,5-Dihydroxy-4-Oxo-1,4-Dihydropyridin-2-Yl)Methoxy]Imino}-N-{(2S)-1-Hydroxy-3-Methyl-3-[(Sulfooxy)Amino]Butan-2-Yl}Ethanamide)
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-05-07 Classification: transferase/transferase inhibitor Ligands: 2U3 |
Organism: Pseudomonas aeruginosa pa1r
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: 2U3
