Search Count: 20
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7F9, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7F9, SO4
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-02-22 Classification: SIGNALING PROTEIN Ligands: 7FX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FX, SO4
 |
Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: TF3, 7F9, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: TF3, 7F9, MG
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FW, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FW, TF3, CL
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FV, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FV, TF3, CL
 |
Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FE, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FE, TF3, CL
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Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: MG, ZZ2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: MG, ZZ2
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Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: DMS, ZZ3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: DMS, ZZ3
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Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: MG, ZZ3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: MG, ZZ3
 |
Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: ZZ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: ZZ4
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Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: ZZ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: ZZ5
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Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: ZZ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: ZZ6
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Orally Active 2-Amino Thienopyrimidine Inhibitors Of The Hsp90 Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-07-28 Classification: CHAPERONE Ligands: 2KL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: 2KL
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4,5 Diaryl Isoxazole Hsp90 Chaperone Inhibitors: Potential Therapeutic Agents For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-12-11 Classification: CHAPERONE Ligands: 2GJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: 2GJ
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4,5 Diaryl Isoxazole Hsp90 Chaperone Inhibitors: Potential Therapeutic Agents For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-12-11 Classification: CHAPERONE Ligands: 2EQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: 2EQ
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Inhibition Of The Hsp90 Molecular Chaperone In Vitro And In Vivo By Novel, Synthetic, Potent Resorcinylic Pyrazole, Isoxazole Amide Analogs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2007-04-24 Classification: CHAPERONE Ligands: MG, SO4, 2GG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-24
Ligands: MG, SO4, 2GG
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3-(5-Chloro-2,4-Dihydroxyphenyl)-Pyrazole-4-Carboxamides As Inhibitors Of The Hsp90 Molecular Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-10-12 Classification: CHAPERONE Ligands: 2D7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-12
Ligands: 2D7
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3-(5-Chloro-2,4-Dihydroxyphenyl)-Pyrazole-4-Carboxamides As Inhibitors Of The Hsp90 Molecular Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2005-10-12 Classification: CHAPERONE Ligands: 2DD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-12
Ligands: 2DD
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Novel, Potent Small Molecule Inhibitors Of The Molecular Chaperone Hsp90 Discovered Through Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2005-06-02 Classification: CHAPERONE Ligands: BSM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-02
Ligands: BSM
 |
Novel, Potent Small Molecule Inhibitors Of The Molecular Chaperone Hsp90 Discovered Through Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-06-02 Classification: CHAPERONE Ligands: CT5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-02
Ligands: CT5