Search Count: 16
![]() |
Structure Of 1 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1P
![]() |
Structure Of 5 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1R
![]() |
Structure Of 10 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.95 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, WYU
![]() |
Structure Of 12 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1Z
![]() |
Structure Of 18 (Bi-2493) In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, VU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, VU6
![]() |
Kras-G12V In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.02 Å Release Date: 2023-06-21 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-21
Ligands: GDP, MG, EDO, OFU
![]() |
Kras In Complex With Precursor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, LR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, LR4
![]() |
Kras In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
![]() |
Kras-G12C In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
![]() |
Kras-G12D In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.09 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
![]() |
Kras-G13D In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
![]() |
Kras-G13D In Complex With Bi-2493
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2023-06-07 Classification: HYDROLASE Ligands: GDP, MG, EDO, VU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, VU6
![]() |
Discovery Of A Kras G12V Inhibitor In Vivo Tool Compound Starting From An Hsqc-Nmr Based Fragment Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-11-09 Classification: SIGNALING PROTEIN Ligands: 2XO, GDP, MG, LX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: 2XO, GDP, MG, LX6
![]() |
Crystal Structure Of Kras-G12C In Complex With Compound 23 (Bi-0474)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXD
![]() |
Crystal Structure Of Kras-G12C In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXK, SO4
![]() |
Crystal Structure Of Bit-Blocked Kras-G12V-S39C In Complex With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, 2XO, MG, LXU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, 2XO, MG, LXU
