Search Count: 16
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Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-05 Classification: Transferase/transferase inhibitor Ligands: 4PV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4PV, GOL
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Pak1 In Complex With 2-Chloro-5-Ethyl-8-Fluoro-11-(4-Methylpiperazin-1-Yl)-Dibenzodiazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OQ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OQ, MG
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Pak1 In Complex With (S)-N-(Tert-Butyl)-3-((2-Chloro-5-Ethyl-8-Fluoro-Dibenzodiazepin-11-Yl)Amino)Pyrrolidine-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OR, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OR, MG
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Crystal Structure Of Renin In Complex With Compound4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2014-10-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 2XF, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: NAG, 2XF, DMS, SO4
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Structure-Based Design Of 4-Hydroxy-3,5-Substituted Piperidines As Direct Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2014-08-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMS, NAG, PO4, 2Y9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: DMS, NAG, PO4, 2Y9
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Crystal Structure Of Renin In Complex With Nvp-Amq838 (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-03-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAG, 0LR
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Crystal Structure Of Renin In Complex With Nvp-Ayz832 (Compound 6A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2013-03-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAG, 0LS, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bca079 (Compound 12A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-03-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAG, 0LT, SO4
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Crystal Structure Of Renin In Complex With Pkf909-724 (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LU, SO4, 0LW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0LU, SO4, 0LW
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Crystal Structure Of Renin In Complex With Gp055321 (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0M2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0M2
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Crystal Structure Of Renin In Complex With Nvp-Ayl747 (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0M3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0M3, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bbv031 (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0ME, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0ME, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bch965 (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0MJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0MJ, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bgq311 (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0N0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0N0, SO4
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Lck Complexed With A Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: 5LK, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: 5LK, EDO
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Human Abl Kinase In Complex With Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2008-04-22 Classification: TRANSFERASE Ligands: NIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NIL