Search Count: 19
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Crystal Structure Of Human Glycine Receptor Alpha-3 Mutant N38Q Bound To Am-3607
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2017-01-18 Classification: TRANSPORT PROTEIN Ligands: 7C6, GLY, ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 7C6, GLY, ZN, CL
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Crystal Structure Of Human Glycine Receptor Alpha-3 Bound To Am-3607
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2017-01-18 Classification: TRANSPORT PROTEIN Ligands: 7C6, GLY, ZN, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 7C6, GLY, ZN, NAG
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B-Raf Wild-Type Kinase Domain In Complex With A Purinylpyridinylamino-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2016-05-04 Classification: Transferase/Transferase Inhibitor Ligands: 5XJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5XJ
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Crystal Structure Of Tankyrase 1 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2C6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: ZN, 2C6
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Co-Crystal Structure Of Tankyrase 1 With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2C8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: ZN, 2C8
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Co-Crystal Structure Of Tankyrase 1 With Compound 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2D6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: ZN, 2D6
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Co-Crystal Structure Of Tankyrase 1 With Compound 2 (5-(2-Aminoquinazolin-6-Yl)-N-(4,4-Dimethyl-2-Oxo-1,2,3,4-Tetrahydroquinolin-7-Yl)-2-Fluorobenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2GU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: ZN, 2GU
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Co-Crystal Structure Of Tankyrase 1 With Compound 3 [(4S)-3-{4-[6-Amino-5-(Pyrimidin-2-Yl)Pyridin-3-Yl]Phenyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One]
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2GV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: ZN, 2GV
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Co-Crystal Structure Of Tankyrase 1 With Compound 4 [(4S)-3-{Trans-4-[6-Amino-5-(Pyrimidin-2-Yl)Pyridin-3-Yl]Cyclohexyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2GY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: ZN, 2GY
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Co-Crystal Structure Of Tnks1 With Compound 52 [N~2-(5-Chloro-2-Methoxyphenyl)-N-[Trans-4-(2-Oxo-2,3-Dihydro-1H-Benzimidazol-1-Yl)Cyclohexyl]Glycinamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-06-05 Classification: Transferase/Transferase Inhibitor Ligands: ZN, K4E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ZN, K4E
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Co-Crystal Structure Of Tnks1 With Compound 18 [4-[(4S)-5,5-Dimethyl-2-Oxo-4-Phenyl-1,3-Oxazolidin-3-Yl]-N-(Quinolin-8-Yl)Benzamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-06-05 Classification: Transferase/Transferase Inhibitor Ligands: ZN, K4F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ZN, K4F
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Crystal Structure Of Ck1G3 With 2-[(4-{[3-(Trifluoromethyl)Pyridin2-Yl]Oxy}Phenyl)Amino]-1H-Benzimidazole-6-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 0VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 0VM
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Crystal Structure Of Ck1G3 With 2-[(4-Tert-Butylphenyl)Amino]-1H-Benzimidazole-6-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 0VN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 0VN
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Crystal Structure Of Tankyrase 1 With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-02-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 1DY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: ZN, 1DY
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Crystal Structure Of Ck1G3 With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-11-21 Classification: transferase/transferase inhibitor Ligands: 0YO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-21
Ligands: 0YO, SO4
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Crystal Structure Of Ck1D With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-11-21 Classification: transferase/transferase inhibitor Ligands: 15G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-21
Ligands: 15G
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Crystal Structure Of Wild Type Braf Kinase Domain In Complex With Organometallic Inhibitor Cns292
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: RSW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-02
Ligands: RSW
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Crystal Structure Of Human Pim1 In Complex With Fluorinated Ruthenium Pyridocarbazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-04-10 Classification: TRANSFERASE Ligands: CL, JM1, EDO, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-10
Ligands: CL, JM1, EDO, EPE
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Crystal Structure Of The Human Pim2 In Complex With A Ruthenium Organometallic Ligand Ru1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2006-08-02 Classification: TRANSFERASE Ligands: HB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-02
Ligands: HB1
