Search Count: 19
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Mcl1 Fab Complex In Complex With Compound 29
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2017-01-18 Classification: IMMUNE SYSTEM Ligands: 7LT |
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 7LT
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Mcl1 Fab Complex In Complex With Compound 21
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2017-01-18 Classification: IMMUNE SYSTEM Ligands: 7LW |
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 7LW
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Crystal Structure Of Mcl1 With Compound 1
Organism: Mus musculus, homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-01-11 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Mus musculus, homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
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Epsp Synthase From Acinetobacter Baumannii
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2016-02-24 Classification: TRANSFERASE |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
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2.37 Angstrom Structure Of Epsp Synthase From Acinetobacter Baumannii
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2016-02-17 Classification: TRANSFERASE Ligands: CL |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2016-02-17
Ligands: CL
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Shikimate Kinase From Acinetobacter Baumannii In Complex With Shikimate
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2015-08-12 Classification: transferase/transferase inhibitor Ligands: SKM, SO4 |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: SKM, SO4
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Crystal Structure Of P. Aeruginosa Ampc
Organism: Pseudomonas aeruginosa (strain atcc 15692 / pao1 / 1c / prs 101 / lmg 12228)
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2015-08-05 Classification: hydrolase/hydrolase inhibitor Ligands: GOL, DMS, 3VT |
Organism: Pseudomonas aeruginosa (strain atcc 15692 / pao1 / 1c / prs 101 / lmg 12228)
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: GOL, DMS, 3VT
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Crystal Structure Of P. Aeruginosa Ampc
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2015-08-05 Classification: hydrolase/hydrolase inhibitor Ligands: GOL, 3VU |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: GOL, 3VU
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Crystal Structure Of P. Aeruginosa Oxa10
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-08-05 Classification: hydrolase/hydrolase inhibitor Ligands: SO4, 3VU, CO2 |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: SO4, 3VU, CO2
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Tmk From S.Aureus In Complex With The Piperidinyl Thymine Class Inhibitor With A C5 Ethyl-Amine
Organism: Staphylococcus aureus (strain mu3 / atcc 700698)
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2015-02-11 Classification: TRANSFERASE Ligands: 43N |
Organism: Staphylococcus aureus (strain mu3 / atcc 700698)
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 43N
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S.Aureus Tmk In Complex With A Potent Inhibitor Compound 18, 2-(3-Chlorophenoxy)-3-Methoxy-4-{[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Methyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 32K |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32K
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S.Aureus Tmk In Complex With Potent Inhibitor Compound 19, 2-(3-Chlorophenoxy)-3-Fluoro-4-{[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Methyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 31Z |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 31Z
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S.Aureus Tmk In Complex With The Potent Inhibitor Compound 38, 2-(3-Chlorophenoxy)-3-Methoxy-4-{(1R)-1-[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Propyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 32B |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32B
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Tmk In Complex With Compound 46, 2-(3-Chlorophenoxy)-3-Fluoro-4-{(1R)-3-Methyl-1-[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Butyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2014-06-11 Classification: Transferase/transferase inhibitor Ligands: 32C |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32C
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S.Aureus Tmk In Complex With Potent Inhibitor Compound 47
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 32E |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32E
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Thymidylate Kinase (Tmk) From S. Aureus In Complex With Tk-666
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0YB |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 0YB
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Crystal Structure Of Thymidylate Kinase From Staphylococcus Aureus Bound To Inhibitor.
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2012-10-24 Classification: Transferase/Transferase inhibitor Ligands: 0Y5 |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 0Y5
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Discovery Of Selective And Potent Inhibitors Of Gram-Positive Bacterial Thymidylate Kinase (Tmk: Compound 41)
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-10-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 13Y |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 13Y
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Discovery Of Selective And Potent Inhibitors Of Gram-Positive Bacterial Thymidylate Kinase (Tmk): Compund 16
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 14D |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 14D
