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14CK image
Structure Of Liver Pyruvate Kinase In Complex With Mitapivat
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, WV2, MG, K

14CL image
Structure Of Liver Pyruvate Kinase In Complex With Tepp-46
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.13 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, 07T, MG, K

14CM image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Site Fragment S3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, WV6, MG, K

14CN image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Site Fragment S4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.93 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, MG, K, WVB

14CO image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Activator 8A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.89 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, WVF, MG, K, EDO

14CP image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Activator 8B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.81 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, WVO, MG, K, EDO

14CQ image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Activator 8C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.18 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, MG, K, WVT

14CR image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Activator 8D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, MG, K, WVX

14CS image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Activator 8E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.13 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, MG, K, WW5, EDO

14CT image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Activator 8F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.48 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, MG, K, WWA

14CU image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Site Binder 8G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.39 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, WWD, MG, K

14CV image
Structure Of Liver Pyruvate Kinase In Complex With Allosteric Site Binder 8H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.07 Å Release Date: 2026-10-14
Classification: TRANSFERASE
Ligands: FBP, OXL, WWI, MG, K

9RN5 image
Crystal Structure Of 33 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2026-08-12
Classification: HYDROLASE
Ligands: A1JR3, MG, ZN

9T3G image
Crystal Structure Of 12 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2026-07-08
Classification: HYDROLASE
Ligands: A1JTA, ZN, MG

9T0T image
Crystal Structure Of The Correct Enantiomer Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2026-05-27
Classification: HYDROLASE
Ligands: A1JS1, A1JS0, MG, ZN

9T1V image
Crystal Structure Of 17 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.41 Å Release Date: 2026-05-27
Classification: HYDROLASE
Ligands: A1JS4, ZN, MG

9T21 image
Crystal Structure Of 29 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.87 Å Release Date: 2026-05-27
Classification: HYDROLASE
Ligands: A1JS7, ZN, MG

7I90 image
Crystal Structure Of 7 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2026-05-20
Classification: HYDROLASE
Ligands: A1B6F, ZN, MG

7I91 image
Crystal Structure Of 13 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.93 Å Release Date: 2026-05-20
Classification: HYDROLASE
Ligands: A1B6S, ZN, MG

7I92 image
Crystal Structure Of 9 Bound To The Ph Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.63 Å Release Date: 2026-05-20
Classification: HYDROLASE
Ligands: A1B6T, ZN, MG
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