Search Count: 18
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Crystal Structure Of Human Monoamine Oxidase B (Mao B) In Complex With 7-[(4-{[(3,4-Dimethoxybenzyl(Methyl)Amino]Methyl}Benzyl)Oxy]-4-(Hydroxymethyl)-2H-Chromen-2-One) (Lp1488)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2026-05-27 Classification: FLAVOPROTEIN Ligands: FAD, A1JF0, C15, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: FAD, A1JF0, C15, GOL
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Recombinant Human Butyrylcholinesterase In Complex With Lp1488 (7-[(4-{[(3,4-Dimethoxybenzyl)(Methyl)Amino]Methyl}Benzyl)Oxy]-4-(Hydroxymethyl)-2H-Chromen-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2026-05-27 Classification: HYDROLASE Ligands: NAG, GOL, MES, SIA, SO4, A1JF0, NA, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: NAG, GOL, MES, SIA, SO4, A1JF0, NA, CL
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Crystal Structure Of Human Soluble Epoxide Hydrolase C-Terminal Domain In Complex With A Benzohomoadamantane-Based Urea Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2025-04-30 Classification: HYDROLASE Ligands: A1H8Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1H8Y
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Crystal Structure Of Tnks2 In Complex With 2-{4-[(2-Hydroxyethyl)(Methyl)Amino]Phenyl}-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: SO4, ZN, 9C5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: SO4, ZN, 9C5, GOL
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Crystal Structure Of Tnks2 In Complex With 2-(2-Aminophenyl)-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: SO4, ZN, 9CE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: SO4, ZN, 9CE, GOL
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Crystal Structure Of Tnks2 In Complex With 2-[4-(4-Methyl-2-Oxoimidazolidin-4-Yl)Phenyl]-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: SO4, ZN, KC8, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: SO4, ZN, KC8, GOL
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Crystal Structure Of Tnks2 In Complex With (5S)-5-Methyl-5-[4-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)Phenyl]Imidazolidine-2,4-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: SO4, F37, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: SO4, F37, ZN
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Crystal Structure Of Tnks2 In Complex With 2-{4-[(2-Hydroxyethyl)(Methyl)Amino]Phenyl}-1,2,3,4-Tetrahydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-21 Classification: TRANSFERASE Ligands: SO4, ZN, 9D5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: SO4, ZN, 9D5, GOL
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Crystal Structure Of Tnks2 In Complex With 2-[4-(Propan-2-Yloxy)Phenyl]-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: SO4, ZN, 9A8, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: SO4, ZN, 9A8, GOL
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Crystal Structure Of Tnks2 In Complex With 2-(3-Hydroxyphenyl)-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: ZN, SO4, 9AN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: ZN, SO4, 9AN, GOL
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Crystal Structure Of Tnks2 In Complex With 2-(4-Ethoxyphenyl)-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: SO4, ZN, 9AQ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: SO4, ZN, 9AQ, GOL
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Crystal Structure Of Tnks2 In Complex With 2-[4-(Pyridin-2-Yl)Phenyl]-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: SO4, ZN, 9AW, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: SO4, ZN, 9AW, GOL
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Crystal Structure Of Tnks2 In Complex With 2-[4-(Piperidin-1-Yl)Phenyl]-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: SO4, ZN, 9B2, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: SO4, ZN, 9B2, GOL, PEG
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Crystal Structure Of Tnks2 In Complex With 2-[4-(Diethylamino)Phenyl]-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: 9C8, ZN, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 9C8, ZN, SO4, GOL
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Crystal Structure Of Tnks2 In Complex With 7-Chloro-2-{4-[(2-Hydroxyethyl)(Methyl)Amino]Phenyl}-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: SO4, ZN, 9CB, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: SO4, ZN, 9CB, GOL
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Crystal Structure Of Tnks2 In Complex With 2-(1H-Indazol-5-Yl)-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-03-07 Classification: TRANSFERASE Ligands: SO4, ZN, 97K, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, ZN, 97K, GOL
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Crystal Structure Of Tnks2 In Complex With 2-(3-Aminophenyl)-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-03-07 Classification: TRANSFERASE Ligands: SO4, ZN, 97H, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, ZN, 97H, GOL
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Crystal Structure Of Tnks2 In Complex With 2-[4-(Morpholin-4-Yl)Phenyl]-3,4-Dihydroquinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-03-07 Classification: HYDROLASE Ligands: ZN, SO4, 97Z, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: ZN, SO4, 97Z, GOL
