Search Count: 21
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Structure Of Sarm1 Tir Domain Bound To G8758
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-02-04 Classification: LYASE Ligands: A1BTS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-04
Ligands: A1BTS
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Structure Of Sarm1 Tir Domain Bound To G6831
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2026-02-04 Classification: LYASE Ligands: A1BU7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-04
Ligands: A1BU7
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Structure Of Sarm1 Tir Domain Bound To G2756
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2026-02-04 Classification: LYASE Ligands: A1BTR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-04
Ligands: A1BTR
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Protac-Induced Ire1 Ternary Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:2.60 Å Release Date: 2025-11-05 Classification: TRANSFERASE Ligands: A1BWF |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-11-05
Ligands: A1BWF
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Human Ebp Complexed With Compound 1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-06-19 Classification: ISOMERASE/INHIBITOR Ligands: A1AEU |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-06-19
Ligands: A1AEU
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Human Ebp Complexed With Compound 3A
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-06-19 Classification: ISOMERASE/INHIBITOR Ligands: A1AEV |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-06-19
Ligands: A1AEV
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Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
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Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: 799 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: 799
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3W
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3R
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3N
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Crystal Structure Of Ire1A In Complex With G-6904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N8S, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N8S, EPE
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Crystal Structure Of Ire1 In Complex With G-3053
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-04-21 Classification: TRANSFERASE/INHIBITOR Ligands: N97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N97
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Crystal Structure Of Ire1A In Complex With G-4100
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
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Structure Of Unphosphorylated Ire1 In Complex With G-1749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJG
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Structure Of Unphosphorylated Ire1 In Complex With G-7658
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJM
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Structure Of Apo Unphosphorylated Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Apo Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Ire1 In Complex With G-0701
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJV
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Structure Of Unphosphorylated Human Ire1 Bound To G-9807
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2020-12-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SJS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJS
