Search Count: 28
 |
Novel Pyrrole Carboxamide Inhibitors Of Jak2 As Potential Treatment Of Myeloproliferative Disorders
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-04-29 Classification: TRANSFERASE Ligands: QUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: QUP
 |
Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: GOL, VVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: GOL, VVQ
 |
Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: 953, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 953, GOL
 |
Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: BJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: BJG
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: H05 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: H05
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: 6LV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: 6LV
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: T62 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: T62
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: TV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: TV2
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: W2D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: W2D
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: HAJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: HAJ
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: G3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: G3R
 |
Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: IK9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: IK9
 |
Structure Of Hsp90 With An Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-10-23 Classification: CHAPERONE Ligands: 50Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-23
Ligands: 50Q
 |
Structure Of Hsp90 With An Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-10-23 Classification: HYDROLASE Ligands: XKL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-23
Ligands: XKL
 |
Structure Of Hsp90 With Nms-E973 Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-05-29 Classification: CHAPERONE Ligands: 9UN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 9UN
 |
Crystal Structure Of Polo-Like Kinase 1 In Complex With A 5-(2-Amino- Pyrimidin-4-Yl)-1H-Pyrrole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: ZN, TLA, 939 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: ZN, TLA, 939
 |
Crystal Structure Of Polo-Like Kinase 1 In Complex With A 2-(2-Amino- Pyrimidin-4-Yl)-1,5,6,7-Tetrahydro-Pyrrolopyridin-4-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: ZN, TLA, 664 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: ZN, TLA, 664
 |
Crystal Structure Of Polo-Like Kinase 1 In Complex With Nms-P937
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-04-06 Classification: TRANSFERASE Ligands: 937, ZN, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: 937, ZN, TLA
 |
Crystal Structure Of Polo-Like Kinase 1 In Complex With A Pyrazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-05-19 Classification: TRANSFERASE Ligands: 071, ZN, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-05-19
Ligands: 071, ZN, TLA
 |
Optimisation Of 6,6-Dimethyl Pyrrolo 3,4-C Pyrazoles: Identification Of Pha-793887, A Potent Cdk Inhibitor Suitable For Intravenous Dosing
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-02-23 Classification: CELL CYCLE Ligands: SO4, 889 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: SO4, 889