Search Count: 19
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1E
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: SO4, A1A1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: SO4, A1A1D
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1C
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1B, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1B, CL
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1A
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Prmt5:Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Prmt5:Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2021-11-17 Classification: Transferase/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
 |
Prmt5:Mep50 Complexed With Adenosine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ADN
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2021-11-17 Classification: transferase/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 10B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: FKY
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 13B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GO7
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 19.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GOD
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: GXA
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Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: WOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: WOE
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: FU5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: FU5
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: FU3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: FU3
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: FU7, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: FU7, PO4
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Crystal Structure Of Human P38Alpha Complexed With A Triazolopyrimidine Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-12-29 Classification: TRANSFERASE Ligands: L9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-29
Ligands: L9G