Search Count: 45
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Bruton'S Tyrosine Kinase (Btk) With Pyridazinone Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2016-09-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, GOL, PG0, 6XL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: SO4, GOL, PG0, 6XL
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Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
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Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
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Egfr Kinase Domain Mutant "Tmlr" With 3-Azetidinyl Azaindazole Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60E
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Cdk8/Cycc In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-04-20 Classification: Transferase/Transcription Ligands: 66X, FMT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 66X, FMT, CL
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Crystal Structure Of Cdk8:Cyclin C Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-02-10 Classification: Transcription/Transferase/Inhibitor Ligands: EDO, FMT, 50R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: EDO, FMT, 50R
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Human Nav1.7-Vsd4-Navab In Complex With Gx-936.
Organism: Arcobacter butzleri, homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.53 Å Release Date: 2015-12-23 Classification: METAL TRANSPORT Ligands: PX4, 5P2 |
Organism: Arcobacter butzleri, homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-23
Ligands: PX4, 5P2
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Egfr Kinase Domain Mutant "Tmlr" With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YV
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Egfr Kinase Domain Mutant "Tmlr" With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YW
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Egfr Kinase Domain Mutant "Tmlr" With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4YX
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Egfr Kinase Domain Mutant "Tmlr" With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4Z8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4Z8
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Egfr Kinase Domain Mutant "Tmlr" With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4ZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4ZB
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Egfr Kinase Domain Mutant "Tmlr" With Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4ZG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4ZG
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Egfr Kinase Domain Mutant "Tmlr" With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4ZH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4ZH
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Egfr Kinase Domain Mutant "Tmlr" With Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4ZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4ZJ
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Egfr Kinase Domain Mutant "Tmlr" With Compound 41A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4ZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4ZQ
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Egfr Kinase Domain Mutant "Tmlr" With Compound 41B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4ZR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4ZR
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Egfr Kinase Domain With Compound 41A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4ZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4ZQ
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Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20J, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20J, PO4, EDO
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Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20M, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20M, PO4, EDO