Search Count: 16
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ7
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ8, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ9
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: Q6K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: Q6K, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations. Compound 51 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1IUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1IUK
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Cd1A-36:2 Sm Binary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2021-05-05 Classification: IMMUNE SYSTEM Ligands: WU7, EDO, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: WU7, EDO, NAG
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Cd1A-42:1 Sm Binary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-05-05 Classification: IMMUNE SYSTEM Ligands: WUA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: WUA, EDO
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Cd1A-42:2 Sm Binary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2021-05-05 Classification: IMMUNE SYSTEM Ligands: FO4, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: FO4, MES
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Crystal Structure Of K103N/Y181C Mutant Hiv-1 Reverse Transcriptase (Rt) In Complex With Idx899
Organism: Human immunodeficiency virus 1, Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2016-02-17 Classification: HYDROLASE Ligands: 5DV |
Organism: Human immunodeficiency virus 1, Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2016-02-17
Ligands: 5DV
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Archaeoglobus Fulgidus Thioredoxin 3 M60H
Organism: Archaeoglobus fulgidus (strain atcc 49558 / vc-16 / dsm 4304 / jcm 9628 / nbrc 100126)
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-04-29 Classification: OXIDOREDUCTASE |
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Rg7109 (N-{4-[6-Tert-Butyl-5-Methoxy-8-(6-Methoxy-2-Oxo-2,5-Dihydropyridin-3-Yl)Quinolin-3-Yl]Phenyl}Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-05-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 28L |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: ZN, 28L
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Compound 48 (N-({(3S)-1-[6-Tert-Butyl-5-Methoxy-8-(2-Oxo-1,2-Dihydropyridin-3-Yl)Quinolin-3-Yl]Pyrrolidin-3-Yl}Methyl)Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-05-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, 28M |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: DMS, 28M
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Crystal Structure Of Jnk1 In Complex With Jip1 Peptide And 7-Fluoro-3-[4-(2-Hydroxy-Ethanesulfonyl)-Benzyl]-4-Oxo-1-Phenyl-1,4-Dihydro-Quinoline-2-Carboxylic Acid Methyl Ester
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: G1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: G1W
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Structure Of Phosphorylated Thr160 Cdk2/Cyclin A In Complex With The Inhibitor Meriolin 3
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-02-12 Classification: TRANSFERASE Ligands: MFR, MG, SGM |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2008-02-12
Ligands: MFR, MG, SGM
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Structure Of Phosphorylated Thr160 Cdk2/Cyclin A In Complex With The Inhibitor Meriolin 5
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-02-12 Classification: TRANSFERASE Ligands: MHR, MG |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2008-02-12
Ligands: MHR, MG
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Structure Of Phosphorylated Thr160 Cdk2/Cyclin A In Complex With The Inhibitor Variolin B
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-02-12 Classification: TRANSFERASE Ligands: VAR, MG, SGM |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2008-02-12
Ligands: VAR, MG, SGM
