Search Count: 58
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Co-Crystal Structure Of Tead1 With Opn-9652
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2025-07-30 Classification: TRANSCRIPTION Ligands: A1H5I, EDO, SO4, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1H5I, EDO, SO4, GOL, PEG
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Crystal Structure Of Gdp-Bound T50I Mutant Of Human Kras4B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-14 Classification: ONCOPROTEIN Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: GDP, MG
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx3397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P31 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: P31
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx8512 In The Dfg-In State
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: WEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: WEG
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx9486 (Bezuclastinib) In The Dfg-In State
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: WEJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: WEJ
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Plx5622
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2019-09-18 Classification: TRANSFERASE Ligands: 622 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-18
Ligands: 622
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N-Terminal Bromodomain Of Brd4 In Complex With Plx5981
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JC
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 6JE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 6JE
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JF
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Crystal Structure Of The Braf (R509H) Kinase Domain Monomer Bound To Vemurafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2016-08-10 Classification: Transferase/Transferase Inhibitor Ligands: 032 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 032
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Crystal Structure Of Braf (R509H) Kinase Domain Bound To Az628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.49 Å Release Date: 2016-08-10 Classification: Transferase/Transferase Inhibitor Ligands: B1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: B1E
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Crystal Structure Of Braf Kinase Domain Bound To Az-Vem
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-08-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6DC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 6DC
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx7904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 904 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 904
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: P06
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx7922
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P02 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: P02
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B-Raf Kinase Domain In Complex With Plx5568
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1OO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 1OO, SO4
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Plx3397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-08-12 Classification: transferase/transferase inhibitor Ligands: P31 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: P31
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Gleevec
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2015-08-12 Classification: transferase/transferase inhibitor Ligands: STI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: STI
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Crystal Structure Of Flt3 With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P30 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: P30
 |
Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx647
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 647 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: 647